Crystal structure of GH71 α-1,3-glucanase Agn1p from<i> Schizosaccharomyces</i><i> pombe:</i> an enzyme regulating cell division in fission yeast, BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 766 151907, 2025.06

Horaguchi, Y; Saitoh, H; Konno, H; Makabe, K; Yano, S

Single Author

Design and Synthesis of Fluorescence-Labeled TAK779 Analogs as Chemical Probes, MOLECULES, 30(12) , 2025.06

Konno, H; Saito, T; Aota, T; Takanuma, D; Okuyama, M; Yokoyama, C

Single Author

Synthesis of Stylissamide B, a Pro-Rich Cyclic Heptapeptide Isolated From the Marine Sponge <i>Stylissa caribica</i>, JOURNAL OF PEPTIDE SCIENCE, 31(6) e70028, 2025.06

Li, YT; Ling, HY; Teruya, K; Konno, H

Single Author

Antifungal activity of GH64 (3-1,3-glucanase from the gram-negative bacterium <i>Flavobacterium johnsoniae</i>, BIOCATALYSIS AND AGRICULTURAL BIOTECHNOLOGY, 66 , 2025.06

Watanabe, A; Yokomichi, M; Suyotha, W; Takahata, Y; Konno, H; Makabe, K; Yano, S

Single Author

Unfolding and refolding of GH19 chitinase Chi19MK with antifungal activity from Lysobacter sp. MK9-1 at low pH and high temperature(タイトル和訳中), Journal of Bioscience and Bioengineering, 139(3) 165-171, 2025.03

Yokomichi Moe, Kanno Haruki, Konno Hiroyuki, Makabe Koki, Yano Shigekazu

Single Author

Unfolding and refolding of GH19 chitinase Chi19MK with antifungal activity from <i>Lysobacter </i>sp. MK9-1 at low pH and high temperature, JOURNAL OF BIOSCIENCE AND BIOENGINEERING, 139(3) 165-171, 2025.03

Yokomichi, M; Kanno, H; Konno, H; Makabe, K; Yano, S

Single Author

Therapeutic effect of curcumin derivative GT863 on prion-infected mice, SCIENTIFIC REPORTS, 15(1) 5444, 2025.02

Teruya, K; Oguma, A; Okuda, M; Iwabuchi, S; Konno, H; Arai, H; Kudo, Y; Sugimoto, H; Doh-ura, K

Single Author

Synthesis and Chemical Structure of the Cyclic Heptapeptide Stylissamide H, JOURNAL OF NATURAL PRODUCTS, 88(2) 593-598, 2025.01

Li, YT; Osanai, S; Nakajima, K; Xu, FS; Sano, H; Sato, H; Katagiri, H; Konno, H

Single Author

Secretoglobin 3A2 peptides have therapeutic potential for allergic airway inflammation, LIFE SCIENCES, 359 123222, 2024.12

Kurotani, R; Sato, Y; Okawara, A; Fukuda, N; Hada, K; Sakahara, S; Takakura, K; Abe, H; Konno, H; Kimura, S

Single Author

Exploring the green synthesis of silver nanoparticles using natural extracts and their potential for cancer treatment, 3 BIOTECH, 14(11) 274, 2024.11

Abdellatif, AAH; Mostafa, MAH; Konno, H; Younis, MA

Single Author

Design of Multi-Target drugs of HDACs and other Anti-Alzheimer related Targets: Current strategies and future prospects in Alzheimer's diseases therapy, BIOORGANIC CHEMISTRY, 151 107651, 2024.10

Soltan, OM; Abdelrahman, KS; Bass, AKA; Takizawa, K; Narumi, A; Konno, H

Single Author

Dynamic Thermodynamic Resolution of Unprotected Amino Acids Using Ni(II) Chiral Schiff Bases, EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 27(36) , 2024.09

Nakano, A; Hayashi, A; Nagaoka, K; Moriwaki, H; Izawa, K; Yano, S; Konno, H

Single Author

Determination of the amino linkage of the D-Dab residue of the cyclic lipo-octapeptide occidiofungins A-D and the antifungal activity of their analogues, ORGANIC & BIOMOLECULAR CHEMISTRY, 22(32) 6575-6581, 2024.08

Kainuma, R; Yano, S; Konno, H

Single Author

Domain structure and function of a-1,3-glucanase Agl-EK14 from the gram-negative bacterium Flavobacterium sp. EK-14, JOURNAL OF BIOSCIENCE AND BIOENGINEERING, 138(2) 118-126, 2024.08

Takahashi, M; Yokomichi, M; Takei, Y; Horaguchi, Y; Makabe, K; Konno, H; Yano, S; Kokeguchi, S

Single Author

Synthesis and evaluation of catecholamine derivatives as amyloid-beta aggregation inhibitors, BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 107 129788, 2024.07

Xu, FS; Takiguchi, Y; Makabe, K; Konno, H

Single Author

Redesign of a thioflavin-T-binding protein with a flat β-sheet to evaluate a thioflavin-T-derived photocatalyst with enhanced affinity, INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 269(Pt 1) 131992, 2024.06

Miura, Y; Namioka, S; Iwai, A; Yoshida, N; Konno, H; Sohma, Y; Kanai, M; Makabe, K

Single Author

SpyTag Peptide with Alkoxyl Aspartic Acids for pH-Dependent Activation of the SpyCatcher/Tag System, BIOCONJUGATE CHEMISTRY, 35(5) 616-622, 2024.04

Che, SJ; Konno, H; Makabe, K

Single Author

Synthesis and Structural Revision of the Cyclic Hexapeptide Dimers Antatollamides A and B, ORGANIC LETTERS, 26(16) 3375-3379, 2024.04

Li, YT; Takamatsu, K; Aota, T; Konno, H

Single Author

Development of 1,5-diarylpyrazoles as EGFR/JNK-2 dual inhibitors: design, synthesis, moleecular docking, and bioactivity evaluation, BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 102 129673, 2024.04

Soltan, OM; Abdel-Aziz, SA; Shaykoon, MS; Osawa, K; Narumi, A; Abdel-Aziz, M; Shoman, ME; Konno, H

Single Author

Addition of α-1,3-glucan-binding domains to α-1,3-glucanase Agn1p from<i> Schizosaccharomyces</i><i> pombe</i> enhances hydrolytic activity of insoluble α-1,3-glucan, JOURNAL OF GENERAL AND APPLIED MICROBIOLOGY, 70(2) 74-81, 2024

Horaguchi, Y; Yokomichi, M; Takahashi, M; Xu, FS; Konno, H; Makabe, K; Yano, S

Single Author

α-1,3-Glucanase from the gram-negative bacterium <i>Flavobacterium</i> sp. EK-14 hydrolyzes fungal cell wall α-1,3-glucan, SCIENTIFIC REPORTS, 13(1) , 2023.12

Takahashi, M; Yano, S; Horaguchi, Y; Otsuka, Y; Suyotha, W; Makabe, K; Konno, H; Kokeguchi, S

Single Author

Synthesis and evaluation of L-dopa and L-Tyr derivatives as amyloid-beta aggregation inhibitors, PHYTOCHEMISTRY LETTERS, 57 239-247, 2023.10

Xu, FS; Okada, M; Makabe, K; Konno, H

Single Author

Heterologous expression of α-1,3-glucanase Agn1p from Schizosaccharomyces pombe, and efficient production of nigero-oligosaccharides by enzymatic hydrolysis from solubilized α-1,3;1,6-glucan, BIOSCIENCE BIOTECHNOLOGY AND BIOCHEMISTRY, 87(10) 1219-1228, 2023.09

Horaguchi, Y; Takahashi, M; Takamatsu, K; Konno, H; Makabe, K; Yano, S

Single Author

Design of the peptide C-terminus protecting group and application for the peptide fragment coupling reaction, TETRAHEDRON LETTERS, 127 , 2023.09

Okawara, A; Hada, K; Kurotani, R; Teruya, K; Konno, H

Single Author

Development and Assessment of 1,5-Diarylpyrazole/Oxime Hybrids Targeting EGFR and JNK-2 as Antiproliferative Agents: A Comprehensive Study through Synthesis, Molecular Docking, and Evaluation, MOLECULES, 28(18) , 2023.09

Abdelrahman, KS; Hassan, HA; Abdel-Aziz, SA; Marzouk, AA; Shams, R; Osawa, K; Abdel-Aziz, M; Konno, H

Single Author

Nigero-oligosaccharide production by enzymatic hydrolysis from alkaline-pretreated a-1,3-glucan, JOURNAL OF BIOSCIENCE AND BIOENGINEERING, 135(3) 182-189, 2023.03

Horaguchi, Y; Yano, S; Takamatsu, K; Otsuka, Y; Suyotha, W; Wakayama, M; Konno, H

Single Author

Structure-Activity Relationship Study of N-Hydroxyphtalimide Derivatives for the Detection of Amines during Fmoc-Solid-Phase Peptide Synthesis, JOURNAL OF ORGANIC CHEMISTRY, 2023.01

Takamatsu, K; Suzuki, R; Matsunaga, A; Katagiri, H; Konno, H

Single Author

Design, Synthesis and Evaluation of Catechol-Based Amyloid Beta Aggregation Inhibitors, HETEROCYCLES, 106(5) 797, 2023

Hiroyuki Konno, Kenta Teruya

Single Author

Antimicrobial Activity of Polysorbate 80-iodine Complex: Polysorbate 80 Firmly Retains Iodine(タイトル和訳中), Journal of Oleo Science, 71(11) 1639-1645, 2022.11

Yano Shigekazu, Terada Senri, Fukushi Misaki, Otsuka Yuitsu, Mizunuma Satomi, Asakura Satoshi, Kawai Takahiro, Konno Hiroyuki, Endo Masatoshi, Nonomura Yoshimune

Single Author

Synthesis and Configuration Confirmation of the ATHOD Fatty Amino Acid Residue in the Burkholdines, JOURNAL OF NATURAL PRODUCTS, 85(8) 2052-2061, 2022.08

Kadowaki, T; Kainuma, R; Kato, S; Konno, H

Single Author

Construction of a fusion protein consisting of α-1,3-glucan-binding domains and tetrameric red fluorescent protein, which is involved in the aggregation of α-1, 3-glucan and inhibition of fungal biofilm formation, JOURNAL OF BIOSCIENCE AND BIOENGINEERING, 133(6) 524-532, 2022.06

Otsuka, Y; Sasaki, K; Suyotha, W; Furusawa, H; Miyazawa, K; Konno, H; Yano, S

Single Author

Design, synthesis, and evaluation of the self-assembled antimicrobial peptides based on the ovalbumin-derived peptide TK913, JOURNAL OF PEPTIDE SCIENCE, 28(4) , 2022.04

Tan, A; Xu, FS; Yokoyama, C; Yano, S; Konno, H

Single Author

Activities of curcumin-related compounds in two cell lines persistently infected with different prion strains, BIOCHIMICA ET BIOPHYSICA ACTA-GENERAL SUBJECTS, 1866(4) , 2022.04

Teruya, K; Iwabuchi, S; Watanabe, Y; Tsuchida, R; Watanabe-Matsui, M; Konno, H; Doh-ura, K

Single Author

APPLICATION OF REVERSIBLE DETECTION METHOD FOR N-TERMINUS AMINO GROUPS: SOLID PHASE SYNTHESIS OF STYLISSATIN B, HETEROCYCLES, 105(1) 397-405, 2022.03

Tan, A; Takamatsu, K; Xu, FS; Osanai, S; Konno, H

Single Author

The Hydrophobicity and Antifungal Potentiation of Burkholdine Analogues, MOLECULES, 27(4) , 2022.02

Konno, H; Sasaki, M; Sano, H; Osawa, K; Nosaka, K; Yano, S

Single Author

New pharmaceuticals approved by FDA in 2020: Small-molecule drugs derived from amino acids and related compounds, CHIRALITY, 34(1) 86-103, 2022.01

Liu, AY; Han, JL; Nakano, A; Konno, H; Moriwaki, H; Abe, H; Izawa, K; Soloshonok, VA

Single Author

Surface Engineering of Top7 to Facilitate Structure Determination, INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 23(2) , 2022.01

Ito, Y; Araki, T; Shiga, S; Konno, H; Makabe, K

Single Author

GH-16 Type β-1,3-Glucanase from<i> Lysobacter</i> sp. MK9-1 Enhances Antifungal Activity of GH-19 Type Chitinase, and Its Glucan-binding Domain Binds to Fungal Cell-wall, JOURNAL OF APPLIED GLYCOSCIENCE, 69(3) 49-56, 2022

Otsuka, Y; Sato, K; Yano, S; Kanno, H; Suyotha, W; Konno, H; Makabe, K; Taira, T

Single Author

Antimicrobial Activity of Polysorbate 80-iodine Complex: Polysorbate 80 Firmly Retains Iodine, JOURNAL OF OLEO SCIENCE, 71(11) 1639-1645, 2022

Yano, S; Terada, S; Fukushi, M; Otsuka, Y; Mizunuma, S; Asakura, S; Kawai, T; Konno, H; Endo, M; Nonomura, Y

Single Author

Synthesis of xylose-binding cyclic octalipopeptides burkholdine-1213 analogues, TETRAHEDRON LETTERS, 87 , 2021.12

Sasaki, M; Kadowaki, T; Kato, S; Chida, S; Yano, S; Nosaka, K; Konno, H

Single Author

Tailor-Made Amino Acids in Pharmaceutical Industry: Synthetic Approaches to Aza-Tryptophan Derivatives, CHEMISTRY-A EUROPEAN JOURNAL, 27(70) 17510-17528, 2021.12

Han, JL; Lyutenko, NV; Sorochinsky, AE; Okawara, A; Konno, H; White, S; Soloshonok, VA

Single Author

Molecular hybrids: A five-year survey on structures of multiple targeted hybrids of protein kinase inhibitors for cancer therapy, EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 225 , 2021.12

Soltan, OM; Shoman, ME; Abdel-Aziz, SA; Narumi, A; Konno, H; Abdel-Aziz, M

Single Author

Nitric oxide protects against ferroptosis by aborting the lipid peroxidation chain reaction, NITRIC OXIDE-BIOLOGY AND CHEMISTRY, 115 34-43, 2021.10

Homma, T; Kobayashi, S; Conrad, M; Konno, H; Yokoyama, C; Fujii, J

Single Author

Comparative study of different chiral ligands for dynamic kinetic resolution of amino acids, CHIRALITY, 33(10) 685-702, 2021.10

Nagaoka, K; Nakano, A; Han, JL; Sakamoto, T; Konno, H; Moriwaki, H; Abe, H; Izawa, K; Soloshonok, VA

Single Author

Carnosine dipeptidase II (CNDP2) protects cells under cysteine insufficiency by hydrolyzing glutathione-related peptides, FREE RADICAL BIOLOGY AND MEDICINE, 174 12-27, 2021.10

Kobayashi, S; Homma, T; Okumura, N; Han, J; Nagaoka, K; Sato, H; Konno, H; Yamada, S; Takao, T; Fujii, J

Single Author

Aerobic oxidation of aldehydes to acids with <i>N</i>-hydroxyphthalimide derivatives, TETRAHEDRON LETTERS, 81 , 2021.09

Takamatsu, K; Kasai, M; Nishizawa, H; Suzuki, R; Konno, H

Single Author

Tailor-made amino acids in the design of small-molecule blockbuster drugs, EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 220 , 2021.08

Han, JL; Konno, H; Sato, T; Soloshonok, VA; Izawa, K

Single Author

Asymmetric Synthesis of α-Difluorinated β-Amino Sulfones through Detrifluoroacetylative Mannich Reactions, EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2021(21) 3035-3038, 2021.06

Li, ZY; Wang, NN; Mei, HB; Konno, H; Soloshonok, VA; Han, JL

Single Author

Asymmetric Synthesis of <i>N</i>-Fmoc-(<i>S</i>)-7-aza-tryptophan via Alkylation of Chiral Nucleophilic Glycine Equivalent, EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2021(21) 2962-2965, 2021.06

Zou, YP; Takeda, R; Han, JL; Konno, H; Moriwaki, H; Abe, H; Izawa, K; Soloshonok, VA

Single Author

Asymmetric synthesis of the two enantiomers of β-phosphorus-containing α-amino acids <i>via</i> hydrophosphinylation and hydrophosphonylation of chiral Ni(ii)-complexes, ORGANIC CHEMISTRY FRONTIERS, 8(10) 2190-2195, 2021.05

Tokairin, Y; Konno, H; Noireau, A; West, C; Moriwaki, H; Soloshonok, VA; Nicolas, C; Gillaizeau, I

Single Author

Production of Chitosanase by <i>Lentzea</i> sp. OUR-I1 Using Acid-Pretreated Shrimp Shell in an Air-Lift Bioreactor and the Feasibility of Utilizing the Residual Biomass, WASTE AND BIOMASS VALORIZATION, 12(5) 2445-2458, 2021.05

Suyotha, W; Cheirsilp, B; Yano, S; Matsuba, S; Konno, H

Single Author

The total synthesis of berberine and selected analogues, and their evaluation as amyloid beta aggregation inhibitors, EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 215 , 2021.04

Tajiri, M; Yamada, R; Hotsumi, M; Makabe, K; Konno, H

Single Author

JNK signaling as a target for anticancer therapy, PHARMACOLOGICAL REPORTS, 73(2) 405-434, 2021.04

Abdelrahman, KS; Hassan, HA; Abdel-Aziz, SA; Marzouk, AA; Narumi, A; Konno, H; Abdel-Aziz, M

Single Author

Cloning, expression, and characterization of a GH 19-type chitinase with antifungal activity from <i>Lysobacter</i> sp. MK9-1, JOURNAL OF BIOSCIENCE AND BIOENGINEERING, 131(4) 348-355, 2021.04

Yano, S; Kanno, H; Tsuhako, H; Ogasawara, S; Suyotha, W; Konno, H; Makabe, K; Uechi, K; Taira, T

Single Author

Maltotriose-Chlorin e6 Conjugate Linked <i>via</i> Tetraethyleneglycol as an Advanced Photosensitizer for Photodynamic Therapy. Synthesis and Antitumor Activities against Canine and Mouse Mammary Carcinoma Cells, ACS OMEGA, 6(10) 7023-7033, 2021.03

Narumi, A; Rachi, R; Yamazaki, H; Kawaguchi, S; Kikuchi, M; Konno, H; Osaki, T; Okamoto, Y; Shen, XD; Kakuchi, T; Kataoka, H; Nomoto, A; Yoshimura, T; Yano, S

Single Author

Asymmetric synthesis of (<i>S</i>)-3-methyleneglutamic acid and its <i>N</i>-Fmoc derivative via Michael addition-elimination reaction of chiral glycine Ni (II) complex with enol tosylates, CHIRALITY, 33(3) 115-123, 2021.03

Shigeno, Y; Han, JL; Soloshonok, VA; Moriwaki, H; Fujiwara, W; Konno, H

Single Author

Design and synthesis of pyrimidine-5-carbonitrile hybrids as COX-2 inhibitors: Anti-inflammatory activity, ulcerogenic liability, histopathological and docking studies, BIOORGANIC CHEMISTRY, 108 , 2021.03

Alfayomy, AM; Abdel-Aziz, SA; Marzouk, AA; Shaykoon, MSA; Narumi, A; Konno, H; Abou-Seri, SM; Ragab, FAF

Single Author

Preparation of SARS-CoV 3CL Protease and Synthesis of its Inhibitors, JOURNAL OF SYNTHETIC ORGANIC CHEMISTRY JAPAN, 79(1) 2-10, 2021.01

Konno, H; Akaji, K

Single Author

Preparation of SARS-CoV 3CL Protease and Synthesis of its Inhibitors, Journal of Synthetic Organic Chemistry, Japan, 79(1) 2-10, 2021

Konno Hiroyuki, Akaji Kenichi

Single Author

PREPARATION OF PYRIDINE DERIVATIVES FROM THE CORRESPONDING 5-ACETAL-1-CARBONYL COMPOUNDS BY ACID PROMOTED CYCLIZATION, HETEROCYCLES, 102(7) 1314-1329, 2021

Mihara, H; Watanabe, Y; Konno, H

Single Author

Peptidomimetics and Peptide-Based Blockbuster Drugs, CURRENT ORGANIC CHEMISTRY, 25(14) 1627-1658, 2021

Han, JL; Konno, H; Sato, T; Izawa, K; Soloshonok, VA

Single Author

Detection of Thiol Functionality and Disulfide Bond Formation by Polyoxometalate, ACS COMBINATORIAL SCIENCE, 22(12) 745-749, 2020.12

Konno, H; Yasumiishi, H; Aoki, R; Nitanai, I; Yano, S

Single Author

Asymmetric synthesis of (<i>S</i>)-α-(octyl)glycine via alkylation of Ni(II) complex of chiral glycine Schiff base, CHIRALITY, 32(12) 1354-1360, 2020.12

Fu, B; Takeda, R; Zou, YPA; Konno, H; Moriwaki, H; Abe, H; Han, JL; Izawa, K; Soloshonok, VA

Single Author

SYNTHESIS AND EVALUATION OF β-GALACTOSIDASE-TARGETING SPIN-LABEL PROBE: 5-<i>O</i>-β-D-GALACTOSYL-5-HYDROXY-1,1,3,3-TETRAMETHYLISOINDOLINE-2-OXYL, HETEROCYCLES, 100(11) 1799-1815, 2020.11

Sugawara, K; Konno, H; Ito, T; Sato, S

Single Author

Design, synthesis and evaluation of diaryl γ-dihydropyrone derivatives as cyclocurcumin mimetics and inhibitors of the aggregation of amyloid β, BIOORGANIC CHEMISTRY, 104 , 2020.11

Hotsumi, M; Tajiri, M; Makabe, K; Konno, H

Single Author

Asymmetric Mannich reactions of (<i>S</i>)-<i>N</i>-<i>tert</i>-butylsulfinyl-3,3,3-trifluoroacetaldimines with yne nucleophiles, BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY, 16 2671-2678, 2020.10

Li, ZY; Wang, L; Huang, YQ; Mei, HB; Konno, H; Moriwaki, H; Soloshonok, VA; Han, JL

Single Author

Antimicrobial activity and secondary structure of a novel peptide derived from ovalbumin, JOURNAL OF PEPTIDE SCIENCE, 26(10) , 2020.10

Tan, A; Suzuki, R; Yokoyama, C; Yano, S; Konno, H

Single Author

Stain Protocol for the Detection of N-Terminal Amino Groups during Solid-Phase Peptide Synthesis, SYNTHESIS-STUTTGART, 52(19) A144-A145, 2020.10

Konno, H; Suzuki, R

Single Author

Stain Protocol for the Detection of N-Terminal Amino Groups-during Solid-Phase Peptide Synthesis, SYNLETT, 31(16) A144-A145, 2020.10

Konno, H; Suzuki, R

Single Author

Tailor-made amino acid-derived pharmaceuticals approved by the FDA in 2019, AMINO ACIDS, 52(9) 1227-1261, 2020.09

Yin, ZZ; Hu, WF; Zhang, W; Konno, H; Moriwaki, H; Izawa, K; Han, JL; Soloshonok, VA

Single Author

Design and Evaluation of Anti-SARS-Coronavirus Agents Based on Molecular Interactions with the Viral Protease, MOLECULES, 25(17) , 2020.09

Akaji, K; Konno, H

Single Author

Residue-Specific Binding Mechanisms of Thioflavin T to a Surface of Flat β-Sheets within a Peptide Self-Assembly Mimic, BIOCHEMISTRY, 59(30) 2782-2787, 2020.08

Namioka, S; Yoshida, N; Konno, H; Makabe, K

Single Author

Synthesis of Ahod Moiety of Ralstonin A Using Amino Acid <i>Schiff</i> Base Ni(II)-Complex Chemistry, HELVETICA CHIMICA ACTA, 103(7) , 2020.07

Oyama, K; Han, J; Moriwaki, H; Soloshonok, VA; Konno, H

Single Author

Michael addition reactions of chiral glycine Schiff base Ni (II)-complex with 1-(1-phenylsulfonyl)benzene, CHIRALITY, 32(6) 885-893, 2020.06

Nagaoka, K; Mei, HB; Guo, YJ; Han, JL; Konno, H; Moriwaki, H; Soloshonok, VA

Single Author

Anti-Alzheimer's flavanolignans from <i>Ceiba pentandra</i> aerial parts, FITOTERAPIA, 143 , 2020.06

Abouelela, ME; Orabi, MAA; Abdelhamid, RA; Abdelkader, MSA; Darwish, FMM; Hotsumi, M; Konno, H

Single Author

Asymmetric Synthesis of Tailor-Made Amino Acids Using Chiral Ni(II) Complexes of Schiff Bases. An Update of the Recent Literature, MOLECULES, 25(12) , 2020.06

Zou, YP; Han, JL; Saghyan, AS; Mkrtchyan, AF; Konno, H; Moriwaki, H; Izawa, K; Soloshonok, VA

Single Author

Stain Protocol for the Detection of N-Terminal Amino Groups during Solid-Phase Peptide Synthesis, ORGANIC LETTERS, 22(9) 3309-3312, 2020.05

Suzuki, R; Konno, H

Single Author

Kitamura Electrophilic Fluorination Using HF as a Source of Fluorine, MOLECULES, 25(9) , 2020.05

Han, JL; Butler, G; Moriwaki, H; Konno, H; Soloshonok, VA; Kitamura, T

Single Author

γ-Glutamylcysteine synthetase and γ-glutamyl transferase as differential enzymatic sources of γ-glutamylpeptides in mice, AMINO ACIDS, 52(4) 555-566, 2020.04

Kobayashi, S; Ikeda, Y; Shigeno, Y; Konno, H; Fujii, J

Single Author

Large-Scale Synthesis of the Glycine Schiff Base Ni(II) Complex Derived from (<i>S</i>)- and (<i>R</i>)-<i>N</i>-(2-Benzoyl-4-chlorophenyl)-1-[(3,4-dichlorophenyl)methyl]-2-pyrrolidinecarboxamide, ORGANIC PROCESS RESEARCH & DEVELOPMENT, 24(2) 294-300, 2020.02

Romoff, TT; Ignacio, BG; Mansour, N; Palmer, AB; Creighton, CJ; Abe, H; Moriwaki, H; Han, JL; Konno, H; Soloshonok, VA

Single Author

Asymmetric Synthesis of 4,4-(Difluoro)glutamic Acid via Chiral Ni(II)-Complexes of Dehydroalanine Schiff Bases. Effect of the Chiral Ligands Structure on the Stereochemical Outcome, CHEMISTRYOPEN, 9(1) 93-96, 2020.01

Tokairin, Y; Shigeno, Y; Han, JL; Roeschenthaler, GV; Konno, H; Moriwaki, H; Soloshonok, VA

Single Author

Synthetic study of cyclic depsipeptide callipeltin Q, Symposium on the Chemistry of Natural Products, symposium papers, 62(0) 313-318, 2020

Tokairin Y., Nagaoka K., Shigeno Y., Gillaizeau I., Soloshonok V., Konno H.

Single Author

Preparative Method for Asymmetric Synthesis of (<i>S</i>)-2-Amino-4,4,4-trifluorobutanoic Acid, MOLECULES, 24(24) , 2019.12

Han, JL; Takeda, R; Liu, XY; Konno, H; Abe, H; Hiramatsu, T; Moriwaki, H; Soloshonok, VA

Single Author

Development of Hamari Ligands for Practical Asymmetric Synthesis of Tailor-Made Amino Acids, ACS OMEGA, 4(21) 18942-18947, 2019.11

Han, JL; Romoff, TT; Moriwaki, H; Konno, H; Soloshonok, VA

Single Author

LC-ESI-MS/MS quantification of carnosine, anserine, and balenine in meat samples, JOURNAL OF CHROMATOGRAPHY B-ANALYTICAL TECHNOLOGIES IN THE BIOMEDICAL AND LIFE SCIENCES, 1132 , 2019.11

Uenoyama, R; Miyazaki, M; Miyazaki, T; Shigeno, Y; Tokairin, Y; Konno, H; Yamashita, T

Single Author

Convenient synthesis of racemic 4,4-difluoro glutamic acid derivatives via Michael-type additions of Ni(II)-complex of dehydroalanine Schiff bases, JOURNAL OF FLUORINE CHEMISTRY, 227 , 2019.11

Tokairin, Y; Soloshonok, VA; Konno, H; Moriwaki, H; Röschenthaler, GV

Single Author

THE ONE-POT SYNTHESIS OF PYRIDINE DERIVATIVES FROM THE CORRESPONDING 1,5-DICARBONYL COMPOUNDS, HETEROCYCLES, 98(10) 1375-1383, 2019.10

Mihara, H; Miyakoshi, T; Kikuchi, Y; Konno, H

Single Author

Design, synthesis, and evaluation of a water soluble C5-monoketone type curcumin analogue as a potent amyloid β aggregation inhibitor, BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 29(16) 2157-2161, 2019.08

Hotsumi, M; Tajiri, M; Nikaido, Y; Sato, T; Makabe, K; Konno, H

Single Author

Quantitative analysis of γ-glutamylpeptides by liquid chromatography-mass spectrometry and application for γ-glutamyltransferase assays, ANALYTICAL BIOCHEMISTRY, 578 13-22, 2019.08

Kobayashi, S; Tokairin, Y; Miyakoshi, T; Saito, T; Nagaoka, K; Ikeda, Y; Fujii, J; Konno, H

Single Author

Antibacterial Activity of 1,2-Alkanediol against <i>Staphylococcus aureus</i> and <i>Staphylococcus epidermidis</i>, JOURNAL OF OLEO SCIENCE, 68(8) 759-763, 2019.08

Okukawa, M; Watanabe, T; Miura, M; Konno, H; Yano, S; Nonomura, Y

Single Author

Low-cost production of chitosanolytic enzymes from <i>Lentzea</i> sp. strain OUR-I1 for the production of antimicrobial substances against food-borne pathogens, INTERNATIONAL FOOD RESEARCH JOURNAL, 26(4) 1293-1304, 2019.08

Huynh, NT; Suyotha, W; Yano, S; Konno, H; Cheirsilp, B; Wakayama, M

Single Author

Synthesis of a burkholdine analogue containing β-hydroxytyrosine, BIOSCIENCE BIOTECHNOLOGY AND BIOCHEMISTRY, 83(7) 1216-1219, 2019.07

Kato, S; Sasaki, M; Yano, S; Konno, H

Single Author

Systematic Analysis of Selective Bactericidal Activity of Fatty Acids against <i>Staphylococcus aureus</i> with Minimum Inhibitory Concentration and Minimum Bactericidal Concentration, JOURNAL OF OLEO SCIENCE, 68(3) 291-296, 2019.03

Watanabe, T; Yamamoto, Y; Miura, M; Konno, H; Yano, S; Nonomura, Y

Single Author

Convergent Synthesis of <i>trans</i>-2,6-Disubstituted Piperidine Alkaloid, (-)-<i>iso</i>-6-Spectaline by Palladium-Catalyzed Cyclization, CHEMICAL & PHARMACEUTICAL BULLETIN, 67(3) 253-257, 2019.03

Kameda, R; Sohma, T; Kobayashi, K; Uchiyama, R; Nosaka, K; Konno, H; Akaji, K; Hattori, Y

Single Author

Thiamin transport in <i>Helicobacter pylori</i> lacking the <i>de novo</i> synthesis of thiamin, MICROBIOLOGY-SGM, 165(2) 224-232, 2019.02

Nosaka, K; Uchiyama, R; Tadano, K; Endo, Y; Hayashi, M; Konno, H; Mimuro, H

Single Author

Improved synthesis of 2,4,6-trialkylpyridines from 1,5-diketoalkanes: total synthesis of anibamine., Org. Biomol. Chem., 17(11) 2896-2905, 2018.12

Miyakoshi, T.; Konno, H.

Multiple Authorship (Including Foreigners)

Convergent synthesis of trans-2,6-disubstituted piperidine alkaloid, (-)-iso-6-spectaline by palladium-catalyzed cyclization., Chem. Pharm. Bull. , 2018.12

79. Kameda, R.; Soma, T.; Kobayashi, K.; Uchiyama, R.; Nosaka, K.; Konno, H.; Akaji, K.; Hattori

Multiple Authorship (Including Foreigners)

Deletion of uncharacterized domain from α-1,3-glucanase of Bacillis circulans KA-304 enhance heterologous enzyme production in Escherichia coli., J. Gen. Appl. Microbiol. , 64(5) 212-220, 2018.11

Yano, S.; Suyotha, W.; Zanma, S.; Konno, H.; Wakamiya, M.

Multiple Authorship (Including Foreigners)

Asymmetric synthesis of (2S,3S)-3-Me-glutamine and (R)-allo-threonine derivatives proper for solid phase peptide coupling., Amino Acids, 51(3) 419-432, 2018.11

Tokairin, Y.; Soloshonok, V. A.; Moriwaki, H.; Konno, H.

Multiple Authorship (Including Foreigners)

Investigation for the cyclization of linear tetrapeptides: Synthesis of tentoxin B and dihydrotentoxin., Tetrahedron, 74(42) 6173-6181, 2018.09

Sato, R.; Oyama, K.; Konno, H.

Multiple Authorship (Including Foreigners)

Design, synthesis and evaluation of curcumin-based fluorescent probes for the detection of A fibrils., Bioorg. Med. Chem. Lett., 28(22) 3520-3525, 2018.09

Sato, T.; Hotsumi, M.; Makabe, K.; Konno, H.

Multiple Authorship (Including Foreigners)

20190820, KAGAKU TO SEIBUTSU, 56(9) 627-634, 2018

KONNO Hiroyuki

Single Author

Synthesis of secretogrobin 3A2 type C (98-139) fragment by Dawson’s native chemical ligation, Tetrahedron Lett. , 58(43) 4145-4148, 2017.10

Kikuchi, M.; Kurotani, R.; Konno, H.

Multiple Authorship (Including Foreigners)

Ralstonins A and B, Lipopeptides with Chlamydospore-Inducing and Phytotoxic Activities from the Plant Pathogen <i>Ralstonia solanacearum</i>, ORGANIC LETTERS, 19(16) 4175-4178, 2017.08

Murai, Y; Mori, S; Konno, H; Hikichi, Y; Kai, K

Single Author

Synthesis and evaluation of phenylisoserine derivatives for the SARS-CoV 3CL protease inhibitor, BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 27(12) 2746-2751, 2017.06

Konno, H; Onuma, T; Nitanai, I; Wakabayashi, M; Yano, S; Teruya, K; Akaji, K

Single Author

Ralstonins A and B, unusual lipopeptides with chlamydospore-inducing and phytotoxic activities from the plant pathogen Ralstonia solanacearum., Org. Lett., 19 4175-4178, 2017.05

Murai, Y.; Mori, S.; Konno H.; Hikichi, Y.; Kai, K.

Multiple Authorship (Including Foreigners)

Synthesis of fully protected (2<i>R,</i>3<i>R,</i>4<i>S)</i>-4-amino-7-guanidino-2,3-dihydroxy heptanoic acid, TETRAHEDRON LETTERS, 58(16) 1604-1606, 2017.04

Yoshino, R; Tokairin, Y; Konno, H

Single Author

Synthesis and evaluation of phenylisoserine derivatives for the SARS-CoV 3CL protease inhibitor., Bioorg. Med. Chem. Lett. , 27 2746-2751, 2017.04

Konno, H.; Onuma, T.; Nitanai, I.; Wakabayashi, M.; Yano, S.; Teruya, K.; Akaji, K.

Multiple Authorship (Including Foreigners)

Synthesis of fully protected (2R,3R,4S)-4-amino-7-guanidino-2,3-dihydroxy heptanoic acid., Tetrahedron Lett. , 58 1604-1606, 2017.03

Yoshino, R.; Tokairin, Y.; Konno, H.

Multiple Authorship (Including Foreigners)

Preparation of (2R,3R,4R)-3-hydroxy-2,4,6-trimethyl heptanoic acid via enzymatic desymmetrization., Tetrahedron, 73 39-45, 2017.02

Tokairin, Y.; Konno, H.

Multiple Authorship (Including Foreigners)

Preparation of (2<i>R</i>, 3<i>R</i>, 4<i>R</i>)-3-hydroxy-2,4,6-trimethylheptanoic acid via enzymatic desymmertization, TETRAHEDRON, 73(1) 39-45, 2017.01

Tokairin, Y; Konno, H

Single Author

Fmoc-OPhth, the reagent of Fmoc protection., Tetrahedron Lett. , 58(16) 1600-1603, 2017.01

Yoshino, R.; Tokairin, Y.; Kikuchi, M.; Konno, H.

Multiple Authorship (Including Foreigners)

Design and synthesis of a series of serine derivatives as small molecule inhibitors of the SARS coronavirus 3CL protease, BIOORGANIC & MEDICINAL CHEMISTRY, 24(6) 1241-1254, 2016.03

Konno, H; Wakabayashi, M; Takanuma, D; Saito, Y; Akaji, K

Single Author

Design and Synthesis of a Series of Serine Derivatives as the Small Molecule Inhibitors of the SARS Coronavirus 3CL Protease., Bioorg. Med. Chem., 24 1241-1254, 2016.03

Konno, H.; Wakabayashi, M.; Takanuma, D.; Saito, Y.; Akaji, K.

Single Author

Synthesis of β-Hydroxytyrosine, A Component of Burkholdines., Nat. Prod. Commun., 11 213-218, 2016.02

Konno, H.; Sasaki, Y.; Sato, R.; Zhu, X.-M.; Otsuki, Y.; Ikoma, M.

Multiple Authorship (Including Foreigners)

Synthesis of β-Hydroxytyrosine, A Component of Burkholdines, NATURAL PRODUCT COMMUNICATIONS, 11(2) 213-218, 2016.02

Konno, H; Sasaki, Y; Sato, R; Zhu, XM; Otsuki, Y; Ikoma, M

Single Author

Cytotoxic evaluation of natural and synthetic callipeltins: a revision of cytotoxicity of callipeltin B., Biosci. Biotechnol. Biochem., 80(6) 1066-1069, 2016.01

Kikuchi, M.; Konno, H.

Multiple Authorship (Including Foreigners)

Synthesis and evaluation of aminopyridine derivatives as potential BACE1 inhibitors, BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 25(22) 5127-5132, 2015.11

Konno, H; Sato, T; Saito, Y; Sakamoto, I; Akaji, K

Single Author

Synthetic study of on homophymine B: solid phase synthesis of a cyclic fragment (vol 56, pg 2809, 2015), TETRAHEDRON LETTERS, 56(31) 4642, 2015.07

Tokairin, Y; Takeda, S; Kikuchi, M; Konno, H

Single Author

Synthetic study of peptide aldehyde via acetal/thioacetal transformation: application for Lys/Ser-containing peptides, TETRAHEDRON, 71(21) 3433-3438, 2015.05

Konno, H; Sema, Y; Tokairin, Y

Single Author

Synthetic study of on homophymine B: solid phase synthesis of a cyclic fragment, TETRAHEDRON LETTERS, 56(21) 2809-2812, 2015.05

Tokairin, Y; Takeda, S; Kikuchi, M; Konno, H

Single Author

Structure activity relationship study of burkholdine analogues toward simple antifungal agents, Bioorg. Med. Chem. Lett., 25(16) 3199-3202, 2015.05

Konno, H.; Abumi, K.; Sasaki, Y.; Yano, S.; Nosaka, K.

Multiple Authorship (Including Foreigners)

Synthetic studies on homophymine B: solid phase synthesis of a cyclic fragment, Tetrahedron Lett. , 56 2809-2812, 2015.04

Tokairin, Y.; Takeda, S.; Kikuchi, M.; Konno, H.

Multiple Authorship (Including Foreigners)

Synthetic study of peptide aldehydes via acetal/thioacetal transformation: application for Lys/Ser-containing peptides, Tetrahedron , 71 3433-3438, 2015.03

Konno, H.; Sema, Y.; Tokairin, Y.

Single Author

Synthesis and evaluation of aminopyridine derivatives as potential BACE1 inhibitors., Bioorg. Med. Chem. Lett. , 25 5127-5132, 2015.02

Konno, H.; Sato, T.; Saito Y.; Sakamoto, I.; Akaji, K.

Multiple Authorship (Including Foreigners)

Synthesis of Orthogonally Protected (2<i>R</i>, 3<i>R</i>, 4<i>S</i>)-4-Amino-2,3-dihydroxyheptane-1,7-dioic Acid, SYNTHESIS-STUTTGART, 47(3) 351-358, 2015.02

Tokairin, Y; Maita, K; Takeda, S; Konno, H

Single Author

Synthesis of orthogonally protected (2R,3R,4S)-4-amino-2,3-dihydroheptan-1,7-dioic acid, Synthesis , 47 351-358, 2015.01

Tokairin, Y.; Maita, K.; Takeda, S.; Konno, H.

Multiple Authorship (Including Foreigners)

Structure activity relationship study of curcumin analogues toward the amyloid-beta aggregation inhibitor, BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 24(24) 5621-5626, 2014.12

Endo, H; Nikaido, Y; Nakadate, M; Ise, S; Konno, H

Single Author

Structure activity relationship study of curcumin analogues toward the amyloid-beta aggregation inhibitor, Bioorg. Med. Chem. Lett., 24 5621-5626, 2014.10

Endo, H.; Nikaido, Y.; Nakadate, M.; Ise, S.; Konno, H.

Multiple Authorship (Including Foreigners)

Total Synthesis of Callipeltin B and M, Peptidyl Marine Natural Products, ORGANIC LETTERS, 16(16) 4324-4327, 2014.08

Kikuchi, M; Konno, H

Single Author

Total synthesis of callipeltin B and M, peptidyl marine natural products, Org. Lett. , 16 4324-4327, 2014.08

Kikuchi, M.; Konno, H.

Multiple Authorship (Including Foreigners)

Effect of prome-site sequence of retro-inverso-modified HTLV-1 protease inhibitor., Bioorg. Med. Chem., 22 2482-2488, 2014.07

Awahara, C.; Tatsumi, T.; Furuta, S.; Shinjoh, G.; Konno, H.; Nosaka, K.; Kobayashi, K.; Hattori, Y.; Akaji, K.

Multiple Authorship (Including Foreigners)

STEREOCHEMICAL ASSIGNMENT OF FOUR DIASTEREOISOMERS OF 3,4-DIMETHYLPYROGLUTAMIC ACID, A MOIETY OF CALLIPELTIN B, HETEROCYCLES, 89(7) 1620-1631, 2014.07

Kikuchi, M; Konno, H

Single Author

Stereochemical assignment of four diastereomers of dimethylpyroglutamic acid, a component of callipeltin B, Heterocycles , 89 1620-1631, 2014.06

Kikuchi, M.; Konno, H.

Single Author

Enzymatic and structural characterization of an archaeal thiamin phosphate synthase., BBA-Proteins and Proteomics, 1844 803-809, 2014.05

Hayashi, M.; Kobayashi, K.; Esaki, H.; Konno, H.; Akaji, K.; Tazuya, K.; Yamada, K.; Nosaka, K.

Multiple Authorship (Including Foreigners)

Effect of prime-site sequence of retro-inverso-modified HTLV-1 protease inhibitor, BIOORGANIC & MEDICINAL CHEMISTRY, 22(8) 2482-2488, 2014.04

Awahara, C; Tatsumi, T; Furuta, S; Shinjoh, G; Konno, H; Nosaka, K; Kobayashi, K; Hattori, Y; Akaji, K

Single Author

Enzymatic and structural characterization of an archaeal thiamin phosphate synthase, BIOCHIMICA ET BIOPHYSICA ACTA-PROTEINS AND PROTEOMICS, 1844(4) 803-809, 2014.04

Hayashi, M; Kobayashi, K; Esaki, H; Konno, H; Akaji, K; Tazuya, K; Yamada, K; Nakabayashi, T; Nosaka, K

Single Author

Synthesis and evaluation of inhibitory activity of the curcumin derivatives toward the inhibitor of beta-site amyloid precursor protein cleaving enzyme 1, Bioorg. Med. Chem. Lett. , 24 685-690, 2014.03

Konno, H.; Endo, H.; Ise, S.; Miyazaki, K.; Aoki, H.; Sanjo, A.; Hattori, Y.; Akaji, K.

Multiple Authorship (Including Foreigners)

Synthetic Study of Callipeltin B: Solid Phase Synthesis and Stereochemical Assignment, Peptide Science 2013, 131-132, 2014.03

Kikuchi, M.; Konno, H.

Multiple Authorship (Including Foreigners)

Synthetic Study on Homophymine A: Stereoselective Synthesis of Unusual Amino Acids and Solid Phase Synthesis of the Cyclic Fragment, Peptide Science 2013, 123-126, 2014.03

Takeda, S.; Tokairin, Y.; Kikuchi, M.; Konno, H.

Multiple Authorship (Including Foreigners)

Synthesis and evaluation of curcumin derivatives toward an inhibitor of beta-site amyloid precursor protein cleaving enzyme 1, BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 24(2) 685-690, 2014.01

Konno, H; Endo, H; Ise, S; Miyazaki, K; Aoki, H; Sanjoh, A; Kobayashi, K; Hattori, Y; Akaji, K

Single Author

Total synthesis of (+)-azimine via diastereoselective aminopalladation, Tetrahedron, 69 8349-8352, 2013.12

Kurogome, Y.; Kosugi, M.; Looi, K. K.; Hattori, Y.; Konno, H.; Hirota, M.; Makabe, H.

Multiple Authorship (Including Foreigners)

Practical synthesis of peptide C-terminal aldehyde on a solid support., Tetrahedron Lett. , 54 4848-4850, 2013.10

Konno, H.; Sema, Y.; Ishii, M.; Hattori, Y.; Nosaka, K.; Akaji, K.

Multiple Authorship (Including Foreigners)

Total synthesis of (+)-azimine via diastereoselective aminopalladation, TETRAHEDRON, 69(39) 8349-8352, 2013.09

Kurogome, Y; Kogiso, M; Looi, KK; Hattori, Y; Konno, H; Hirota, M; Makabe, H

Single Author

Practical synthesis of peptide C-terminal aldehyde on a solid support, TETRAHEDRON LETTERS, 54(36) 4848-4850, 2013.09

Konno, H; Sema, Y; Ishii, M; Hattori, Y; Nosaka, K; Akaji, K

Single Author

Improved synthesis of D-allothreonine derivatives from L-threonine, TETRAHEDRON, 69(34) 7098-7101, 2013.08

Kikuchi, M; Konno, H

Single Author

Synthesis and antifungal activities of cyclic octa-lipopeptide burkholdine analogues, Bioorg. Med. Chem. Lett. , 23 4244-4247, 2013.08

Konno, H.; Otsuki, Y.; Matsuzaki, K.; Nosaka, K.

Multiple Authorship (Including Foreigners)

Synthesis and antifungal activities of cyclic octa-lipopeptide burkholdine analogues, BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 23(14) 4244-4247, 2013.07

Konno, H; Otsuki, Y; Matsuzaki, K; Nosaka, K

Single Author

Improved synthesis of D-allothreonine derivatives from L-threonine, Tetrahedron , 69 7098-7101, 2013.06

Kikuchi, M.; Konno, H.

Multiple Authorship (Including Foreigners)

Education project for Innovation, Executed in Faculty of Engineering at Yamagata University in 2010 –Two Education programs about biomass and snow vehicle-, J. Engineering Edu. Res, 14 21-29, 2012.10

Furukawa, H.; Watanabe, K.; Konno, H.; Matsushima, Y.; Matsuba, G.; Nomoto, K.

Multiple Authorship (Including Foreigners)

Synthesis and evaluation of SARS 3CL protease inhibitors using the serine template, Proceedings of 32nd European Peptide Symposium, 478-479, 2012.10

Takanuma, D.; Akaji, K.; Konno, H.

Multiple Authorship (Including Foreigners)

Synthesis of cyclic lipo-peptide derivatives of burkholdines and its antifungal activity, Proceedings of 32nd European Peptide Symposium, 80-81, 2012.10

Konno, H.; Otsuki, Y.

Multiple Authorship (Including Foreigners)

Synthetic study of callipeltin B analogues and its cytotoxicity, Proceedings of 32nd European Peptide Symposium, 636-637, 2012.10

Kikuchi, M.; Watanabe, Y.; Tanaka, M.; Akaji, K.; Konno, H.

Multiple Authorship (Including Foreigners)

Synthesis and Evaluation of SARS 3CL Protease Inhibitors Using the Serine Template, JOURNAL OF PEPTIDE SCIENCE, 18 S148, 2012.09

Takanuma, D; Akaji, K; Konno, H

Single Author

Synthesis of cyclic lipo-octapeptide derivatives of burkholdines and its antifungal activity, JOURNAL OF PEPTIDE SCIENCE, 18 S43, 2012.09

Konno, H; Otsuki, Y

Single Author

Synthetic Study of Callipeltin B Analogues and its Cytotoxicity, JOURNAL OF PEPTIDE SCIENCE, 18 S189-S190, 2012.09

Kikuchi, M; Watanabe, Y; Tanaka, M; Akaji, K; Konno, H

Single Author

Synthesis of Bioactive Natural Products as Protein Inhibitors, BIOSCIENCE BIOTECHNOLOGY AND BIOCHEMISTRY, 76(7) 1257-1261, 2012.07

Konno, H

Single Author

Facilitated recruitment of Pdc2p, a yeast transcriptional activator, in response to thiamin starvation, FEMS Microbiol. Lett. , 330 140-147, 2012.06

Nosaka, K.; Esaki, H.; Onozuka, M.; Konno, H.; Hattori, Y.; Akaji, K.

Multiple Authorship (Including Foreigners)

Facilitated recruitment of Pdc2p, a yeast transcriptional activator, in response to thiamin starvation, FEMS MICROBIOLOGY LETTERS, 330(2) 140-147, 2012.05

Nosaka, K; Esaki, H; Onozuka, M; Konno, H; Hattori, Y; Akaji, K

Single Author

Structure-Based Design, Synthesis, and Evaluation of Peptide-Mimetic SARS 3CL Protease Inhibitors, JOURNAL OF MEDICINAL CHEMISTRY, 54(23) 7962-7973, 2011.12

Akaji, K; Konno, H; Mitsui, H; Teruya, K; Shimamoto, Y; Hattori, Y; Ozaki, T; Kusunoki, M; Sanjoh, A

Single Author

Structure-Based Design, Synthesis, and Evaluation of Peptide-mimetics SARS 3CL Protease Inhibitors, J. Med. Chem. , 54 7962-7973, 2011.12

Akaji, K.; Konno, H.; Mitsui H.; Teruya, K.; Hattori, Y.; Ozaki, T.; Kusunoki, M.; Sanjho, A.

Multiple Authorship (Including Foreigners)

Synthesis of tokaramide A, a cysteine protease inhibitor from marine sponge <i>Theonella aff</i>. <i>mirabilis</i>, TETRAHEDRON, 67(47) 9067-9071, 2011.11

Konno, H; Nosaka, K; Akaji, K

Single Author

Synthesis and cytotoxicity of the depsipeptides analogues of callipeltin B, BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 21(16) 4865-4868, 2011.08

Kikuchi, M; Watanabe, Y; Tanaka, M; Akaji, K; Konno, H

Single Author

Solid phase total synthesis of callipeltin E isolated from marine sponge <i>Latrunculia</i> sp., TETRAHEDRON LETTERS, 52(30) 3872-3875, 2011.07

Kikuchi, M; Nosaka, K; Akaji, K; Konno, H

Single Author

Synthesis of N1- and N8-(γ-L-Glutamyl)spermidines and (γ-L-Glutamyl)putrescine. , Lett. In Org. Chem., 8 1-5, 2011.04

Toho, K.; Abe, N.; Yamada, T.; the late Ito, Y.; Konno, H.; Kuwahara, S.; Kiyota, H.

Multiple Authorship (Including Foreigners)

Synthesis of tokaramide A, a cysteine protease inhibitor from marine sponge Theonella mirabilis., Konno, H.; Nosaka, K.; Akaji, K., 67 9067-9071, 2011.04

Konno, H.; Nosaka, K.; Akaji, K.

Multiple Authorship (Including Foreigners)

Synthesis and cytotoxicity of callipeltin B analogues., Bioorg. Med. Chem. Lett., 21 4865-4868, 2011.04

Kikuchi, M.; Watanabe, Y; Tanaka, M.; Akaji, K.; Konno, H.

Multiple Authorship (Including Foreigners)

Solid Phase Total Synthesis of Callipeltin E isolated from marine sponge Latrunculia sp., Tetrahedron Lett. , 52(30) 3872-3875, 2011.04

Kikuchi, M.; Nosaka, K.; Akaji, K.; Konno, H.

Multiple Authorship (Including Foreigners)

Synthesis of Annonaceous Acetogenins and Their Inhibitory Action with Mitochondrial Complex I, JOURNAL OF SYNTHETIC ORGANIC CHEMISTRY JAPAN, 69(2) 159-168, 2011.02

Hattori, Y; Konno, H; Miyoshi, H; Makabe, H

Single Author

Synthesis of <i>N<SUP>1</SUP></i>- and <i>N<SUP>8</SUP></i>-(γ-L-Glutamyl)spermidines and (γ-L-Glutamyl) putrescine, LETTERS IN ORGANIC CHEMISTRY, 8(1) 1-4, 2011.01

Toho, K; Abe, N; Yamada, T; Ito, Y; Konno, H; Kuwahara, S; Kiyota, H

Single Author

Synthesis of solamin type mono-THF acetogenins using cross-metathesis, TETRAHEDRON, 66(40) 7946-7953, 2010.10

Konno, H; Makabe, H; Hattori, Y; Nosaka, K; Akaji, K

Single Author

Synthesis of Annonacin Isolated from <i>Annona densicoma</i>, BIOSCIENCE BIOTECHNOLOGY AND BIOCHEMISTRY, 74(6) 1274-1275, 2010.06

Oasa, M; Hattori, Y; Konno, H; Makabe, H

Single Author

Synthetic Studies on Callipeltins: stereoselective syntheses of (3S, 4R)-3,4-dimethyl-L-pyroglutamic acid and Fmoc-D-allothreonine., Heterocycles, 81(1) 79-89, 2010.04

Konno, H.; Takebayashi, Y.; Nosaka, K.; Akaji, K.

Multiple Authorship (Including Foreigners)

Synthesis of solamin type mono-THF acetogenins using cross-metathesis, Tetrahedron , 66 7946-7953, 2010.04

Konno, H.; Makabe, H.; Yattori, Y.; Nosaka, K.; Akaji, K.

Multiple Authorship (Including Foreigners)

Synthesis of Annonacin, Biosci. Biotetcnol. Biochem. , 76(4) 1274-1275, 2010.04

Oasa, M.; Hattori, Y.; Konno, H.; Makabe, H.

Multiple Authorship (Including Foreigners)

Evaluation of retro-inverso modifications of HTLV-1 protease inhibitors containing a hydroxyethylamine isoster., Bioorg. Med. Chem., 18 2720-2727, 2010.04

Tatsumi, T.; Awahara, C.; Naka, H.; Aimoto, S.; Konno, H.; Nosaka, K.; Akaji, K.

Multiple Authorship (Including Foreigners)

Evaluation of retro-inverso modifications of HTLV-1 protease inhibitors containing a hydroxyethylamine isoster, BIOORGANIC & MEDICINAL CHEMISTRY, 18(7) 2720-2727, 2010.04

Tatsumi, T; Awahara, C; Naka, H; Aimoto, S; Konno, H; Nosaka, K; Akaji, K

Single Author

SYNTHETIC STUDIES ON CALLIPELTINS: STEREOSELECTIVE SYNTHESES OF (3<i>S</i>,4<i>R</i>)-3,4-DIMETHYL-L-PYROGLUTAMIC ACID AND FMOC-D-ALLOTHREONINE FROM SERINE DERIVATIVES, HETEROCYCLES, 81(1) 79-89, 2010.01

Konno, H; Takebayashi, Y; Nosaka, K; Akaji, K

Single Author

A CONCISE SYNTHESIS OF SOLAMIN AND <i>CIS</i>-SOLAMIN, MONO-THF ACETOGENINS FROM <i>ANNONA MURICATA</i>, HETEROCYCLES, 78(9) 2369-2376, 2009.09

Makabe, H; Kuwabara, A; Hattori, Y; Konno, H

Single Author

Synthesis of [19, 35, 36-<SUP>13</SUP>C₃]-labeled TAK779 as a molecular probe, BIOORGANIC & MEDICINAL CHEMISTRY, 17(16) 5769-5774, 2009.08

Konno, H; Aimoto, S; Smith, SO; Nosaka, K; Akaji, K

Single Author

Evaluation of Lipid-Binding Propaties of the N-Terminal Helical Segments in Human Apolipoprotein A-I Using Fragment Peptides, J. Peptide Sci. , 15(1) 36-42, 2009.04

Tanaka, M.; Tanaka, T.; Ohta, S.; Kawakami, T.; Konno, H.; Akaji, K.; Aimoto, S.; Saito, H.

Multiple Authorship (Including Foreigners)

Synthesis of [19.35.36-13C3]-Labeled TAK779 as a moleculer probe, Bioorg. Med. Chem., 17 5769-5774, 2009.04

Konno, H.; Aimoto, S.; Smith, S. O.; Nosaka, K.; Akaji, K.

Multiple Authorship (Including Foreigners)

A Concise Synthesis of Solamin and cis-Solamin, Mono-THF Acetogenins from Annona muricata, Heterocycles, 78(9) 2369-2376, 2009.04

Makabe, H.; Kuwabara, A.; Hattori, Y.; Konno, H.

Multiple Authorship (Including Foreigners)

Evaluation of lipid-binding properties of the N-terminal helical segments in human apolipoprotein A-I using fragment peptides, JOURNAL OF PEPTIDE SCIENCE, 15(1) 36-42, 2009.01

Tanaka, M; Tanaka, T; Ohta, S; Kawakami, T; Konno, H; Akaji, K; Aimoto, S; Saito, H

Single Author

Thiamin-dependent transactivation activity of <i>PDC2</i> in <i>Saccharomyces cerevisiae</i>, FEBS LETTERS, 582(29) 3991-3996, 2008.12

Nosaka, K; Onozuka, M; Konno, H; Akaji, K

Single Author

Evaluation of peptide-aldehyde inhibitors using R188I mutant of SARS 3CL protease as a proteolysis-resistant mutant, BIOORGANIC & MEDICINAL CHEMISTRY, 16(21) 9400-9408, 2008.11

Akaji, K; Konno, H; Onozuka, M; Makino, A; Saito, H; Nosaka, K

Single Author

Synthesis of pyranicin and its deoxygenated analogues and their inhibitory action with bovine heart mitochondrial complex I, TETRAHEDRON, 64(33) 7695-7703, 2008.08

Furuhata, S; Hattori, Y; Okajima, M; Konno, H; Abe, M; Miyoshi, H; Goto, T; Makabe, H

Single Author

Synthesis of pyranicin and its inhibitory action with bovine heart mitochondrial complex I, ORGANIC LETTERS, 10(5) 717-720, 2008.03

Hattori, Y; Furuhata, S; Okajima, M; Konno, H; Abe, M; Miyoshi, H; Goto, T; Makabe, H

Single Author

Involvement of thiaminase II encoded by the <i>THI20</i> gene in thiamin salvage of <i>Saccharomyces cerevisiae</i>, FEMS YEAST RESEARCH, 8(2) 266-275, 2008.03

Onozuka, M; Konno, H; Kawasaki, Y; Akaji, K; Nosaka, K

Single Author

Total synthesis of <i>cis</i>-solamin A, a mono-tetrahydrofuran acetogenin isolated from <i>Annona muricata</i>, TETRAHEDRON LETTERS, 49(5) 782-785, 2008.01

Konno, H; Okuno, Y; Makabe, H; Nosaka, K; Onishi, A; Abe, Y; SUgirnoto, A; Akaji, K

Single Author

Possible involvement of thiaminase II encoded by the THI20 gene in thiamine salvage of Saccharomyces cerevisiae, Journal of FEMS Yeast Research, 8(2) 266-275, 2008.01

Onozuka, M.; Konno, H.; Kawasaki, Y.; Akaji, K.; Nosaka, K.

Multiple Authorship (Including Foreigners)

Synthesis of Pyranicin and its Inhibitory Action with Bovine Heart Mitochondrial Complex I, Organic Letters, 10(5) 717-720, 2008.01

Hattori, N.; Furuhata, S.; Okajima, M.; Konno, H.; Abe, M.; Miyoshi, H.; Goto, T, Makabe, H.

Multiple Authorship (Including Foreigners)

Total synthesis of pyranicin and its deoxygenated analogues and their inhibitory action with bovine heart mitochondrial complex I, Tetrahedron, 64 7695-7703, 2008.01

Furuhata, S.; Hattori, Y.; Okajima, M.; Konno, H.; Abe, M.; Miyoshi, H.; Goto, T.; Makabe, H.

Multiple Authorship (Including Foreigners)

Thiamin-dependent transactivation activity of PDC2 in Saccharomyces, FEBS Letters, 582(29) 3991-3996, 2008.01

Nosaka, K.; Onozuka, M.; Konno, H.; Akaji, K.

Multiple Authorship (Including Foreigners)

Evaluation of Peptide Aldehyde Inhibitors using R188I Mutant of SARS 3CL Protease as a proteolysis-resistant mutant, Bioorganic Medicinal Chemistry, 16 9400-9408, 2008.01

Akaji, K.; Konno, H.; Onozuka, M.; Makino, A.; Nosaka, K.

Multiple Authorship (Including Foreigners)

Total synthesis of cis-solamin A, a mono-tetrahydrofuran acetogenin isolated from Annona muricata. , Tetrahedron Letters, 49(5) 782-785, 2008.01

Konno, H.; Okuno, Y.; Makabe, H.; Nosaka, K.; Onishi, A.; Abe, N.; Sugimoto, A.; Akaji, K.

Multiple Authorship (Including Foreigners)

Stereoselective synthesis of β-methoxytyrosine derivatives for identification of the absolute configuration of callipeltin E, SYNTHESIS-STUTTGART, (23) 3666-3672, 2007.12

Konno, H; Aoyama, S; Nosaka, K; Akaji, K

Single Author

Synthesis of All Stereoisomers of β-Methoxy Tyrosine Derivatives and Identification of the Absolute Configration in Callipeltin E, Synthesis, (23) 3666-3672, 2007.12

Konno, H.; Aoyama, S.; Nosaka, K.; Akaji, K.

Multiple Authorship (Including Foreigners)

Total Synthesis of Miraziridine A and Identification of Its Major Reactive Site for Cathepsin B, Tetrahedron, 63(38) 9502-9513, 2007.10

Konno, H.; Kubo, K.; Makabe, H.; Toshiro, E.; Nosaka, K.; Akaji, K.

Multiple Authorship (Including Foreigners)

Total synthesis of miraziridine A and identification of its major reaction site for cathepsin B, TETRAHEDRON, 63(38) 9502-9513, 2007.09

Konno, H; Kubo, K; Makabe, H; Toshiro, E; Hinoda, N; Nosaka, K; Akaji, K

Single Author

Studies on Substrate Specificity at PR/p3 Cleavage Site of HTVL-1 Protease, Int. J. Peptide Res., 13 173-179, 2007.08

Bang, J. K.; Teruya, K.; Aimoto, S.; Konno, H.; Nosaka, K.; Tatsumi, T.; Akaji, K.

Multiple Authorship (Including Foreigners)

Total Synthesis of Miraziridine A and Its Analogues, Peptides, 1-2, 2007.08

Konno, H.; Kubo, K.; Makabe, H.; Nosaka, K.; Akaji, K.

Multiple Authorship (Including Foreigners)

Studies on substrate specificity at PR/p3 cleavage site of HTLV-1 protease, INTERNATIONAL JOURNAL OF PEPTIDE RESEARCH AND THERAPEUTICS, 13(1-2) 173-179, 2007.06

Bang, JK; Teruya, K; Aimoto, S; Konno, H; Nosaka, K; Tatsumi, T; Akaji, K

Single Author

Synthesis, determination of the absolute configuration of tonkinelin, and inhibitory action with bovine heart mitochondrial complex I, BIOORGANIC & MEDICINAL CHEMISTRY, 15(8) 3026-3031, 2007.04

Hattori, Y; Konno, H; Abe, M; Miyoshi, H; Goto, T; Makabe, H

Single Author

Synthesis of (17S, 18S)- and (17R, 18R)-tonkinelin and their inhibitory action with bovine heart mitochondorial complex I, Bioorg. Med. Chem. , 15 3026-3031, 2007.04

Hattori, Y.; Konno, H.; Abe, M.; Miyoshi, H.; Goto, T.; Makabe, H.

Multiple Authorship (Including Foreigners)

First syntheses of Trans- and Cis-dendrochrysanines, Heterocycles, 68(12) 2579-2585, 2006.12

Konno, H.; Kusumoto, S.; Kanai, S.; Yamahana, Y.; Nosaka, K.; Akaji, K.

Multiple Authorship (Including Foreigners)

First synthesis of <i>trans</i>- and <i>cis</i>-dendrochrysanines, HETEROCYCLES, 68(12) 2579-2585, 2006.12

Konno, H; Kusumoto, S; Kanai, S; Yamahana, Y; Nosaka, K; Akaji, K

Single Author

Synthesis of murisolin, (15<i>R</i>, 16<i>R</i>, 19<i>R</i>, 20<i>S</i>)-murisolin A, and (15<i>R</i>, 16<i>R</i>, 19<i>S</i>, 20<i>S</i>)-16,19-<i>cis</i>-murisolin and their inhibitory action with bovine heart mitochondrial complex I, CHEMISTRY-AN ASIAN JOURNAL, 1(6) 894-904, 2006.12

Hattori, Y; Kimura, Y; Moroda, A; Konno, H; Abe, M; Miyoshi, H; Goto, T; Makabe, H

Single Author

Synthesis of Murisolin, (15R, 16R, 19R, 20S)-Murisolin-A, (15R, 16R, 19R, 20S)-16,19-cis-Murisolin-A, and Their Inhibitory Action with Bovine Heart Mitochondrial Complex I, Chemistry-Asian Journal , 1 894-904, 2006.11

Hattori, Y.; Kimura, Y.; Moroda, A.; Konno, H.; Abe, M.; Miyoshi, H.; Goto, T, Makabe, H.

Single Author

Evaluations of Substrate Specificity and Inhibition at PR/p3 Cleavage Site of HTLV-1 Protease, Bioorg. Med. Chem. Lett. , 16 3761-3764, 2006.10

Naka, H.; Teruya, K.; Bang, J. K.; Aimoto, S.; Tatsumi, T.; Konno, H.; Nosaka, K.; Akaji, K.

Multiple Authorship (Including Foreigners)

Synthesis of (4R, 15R, 16R, 21S)-and (4R, 15S, 16S, 21S)-rollicosin and squamostolide, and their inhibitory action with bovine heart mitochondeial complex I, Bioorg. Med. Chem. Lett. , 14 3119-3130, 2006.09

22. Makabe, H.; Kimura, Y.; Higuchi, M.; Konno, H.; Murai, M.; Miyoshi, H.

Multiple Authorship (Including Foreigners)

Evaluations of substrate specificity and inhibition at PR/p3 cleavage site of HTLV-1 protease, BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 16(14) 3761-3764, 2006.07

Naka, H; Teruya, K; Bang, JK; Aimoto, S; Tatsumi, T; Konno, H; Nosaka, K; Akaji, K

Single Author

Synthetic Studies on Miraziridine A, a Cysteine Protease Inhibitor Isolated from Theonella aff. mirabilis., Proceedings of 43JPS/PEM4, 37-38, 2006.05

Konno, H.; Kubo, K.; Makabe, H.; Nosaka, K.; Akaji, K.

Multiple Authorship (Including Foreigners)

Synthesis of (4<i>R</i>,15<i>R</i>,16<i>R</i>,21<i>S</i>)- and (4<i>R</i>,15<i>S</i>,16<i>S</i>,21<i>S</i>)-rollicosin, squamostolide, and their inhibitory action with bovine heart mitochondrial complex I, BIOORGANIC & MEDICINAL CHEMISTRY, 14(9) 3119-3130, 2006.05

Makabe, H; Kimura, Y; Higuchi, M; Konno, H; Murai, M; Miyoshi, H

Single Author

Solid-phase syntheses of olefin-containing inhibitors for HTLV-1 protease using the Horner-Emmons reaction, JOURNAL OF ORGANIC CHEMISTRY, 70(25) 10596-10599, 2005.12

Bang, JK; Naka, H; Teruya, K; Aimoto, S; Konno, H; Nosaka, K; Tatsumi, T; Akaji, K

Single Author

Solid-Phase Synthesis of Olefin-containing Inhibitors for HTLV-1 Protease using the Horner-Emmons Reaction, J. Org. Chem., 70 10596-10599, 2005.12

Bang, J. K.; Naka, H.; Teruya, K.; Aimoto, S.; Konno, H.; Nosaka, K.; Akaji, K.

Multiple Authorship (Including Foreigners)

Genetic regulation mediated by thiamin pyrophosphate-binding motif in Saccharomyces cerevisiae, Mol. Microbiol., 58 467-479, 2005.11

Nosaka, K.; Onozuka, M.; Konno, H.; Kawasaki, Y.; Nishino, H.; Sano, M.; Akaji, K.

Multiple Authorship (Including Foreigners)

Molecular Cloning and Analysis of the 5’-Flanking Region of the Human Thiamin Pyrophosphokinase gene, J. Nutr. Sci. Vitaminol. , 51 274-277, 2005.10

Onozuka, M.; Konno, H.; Akaji, K.; Nishino, H.; Nosaka, K.

Multiple Authorship (Including Foreigners)

Genetic regulation mediated by thiamin pyrophosphate-binding motif in <i>Saccharomyces cerevisiae</i>, MOLECULAR MICROBIOLOGY, 58(2) 467-479, 2005.10

Nosaka, K; Onozuka, M; Konno, H; Kawasaki, Y; Nishimura, H; Sano, M; Akaji, K

Single Author

Synthesis of (4R, 15R, 16R, 21S)-and (4R, 15S, 16S, 21S)-rollicosin and squamostolide, and their inhibitory action with bovine heart mitochondeial complex I, Tetrahedron Lett. , 46 4671-4675, 2005.09

Makabe, H.; Higuchi, M.; Konno, H.; Murai, M.; Miyoshi, H.

Multiple Authorship (Including Foreigners)

Genetic Regulation Mediated by Thiamin Pyrophosphate-binding Motif in Saccharomyces cerevisiae. , Proceeding of the XXIInd International Conference on Yeast Genetics &Molecular Biology, -22, 2005.08

Nosaka, K.; Onozuka, M.; Kawasaki, Y.; Konno, H.; Akaji, K.

Multiple Authorship (Including Foreigners)

Molecular cloning and analysis of the 5′-fanking region of the human thiamin pyrophosphokinase, JOURNAL OF NUTRITIONAL SCIENCE AND VITAMINOLOGY, 51(4) 274-277, 2005.08

Onozuka, M; Konno, H; Akaji, K; Nishino, H; Nosaka, K

Single Author

Synthesis of (4<i>R</i>,15<i>R</i>,16<i>R</i>,21<i>S</i>)- and (4<i>R</i>,15<i>S</i>,16<i>S</i>,21<i>S</i>)-rollicosin, TETRAHEDRON LETTERS, 46(27) 4671-4675, 2005.07

Makabe, H; Higuchi, M; Konno, H; Murai, M; Miyoshi, H

Single Author

Total Synthesis of cis-Solamin and Its Inhibitory Action with Mitochondrial Complex I, Tetrahedron Lett. , 60 10651-10657, 2004.12

Makabe, H.; Hattori, Y.; Kimura, Y.; Konno, H.; Abe, M.; Miyoshi, H.; Tanaka, A.; Oritani, T.

Multiple Authorship (Including Foreigners)

Total synthesis of <i>cis</i>-solamin and its inhibitory action with bovine heart mitochondrial complex I, TETRAHEDRON, 60(47) 10651-10657, 2004.11

Makabe, H; Hattori, Y; Kimura, Y; Konno, H; Abe, M; Miyoshi, H; Tanaka, A; Oritani, T

Single Author

Synthesis of Two Possible Diastereoisomers of Reticulatain-1, Tetrahedron Lett. , 45 973-977, 2004.11

Makabe, H.; Miyawaki, A.; Takahashi, R.; Hattori, Y.; Konno, H.; Abe, M.; Miyoshi, H.

Multiple Authorship (Including Foreigners)

Synthesis and Mitochondrial Inhibition of Dihydroxy-Cohibin A, Non-THF Annonaceous Acetogenin Analogue, Bioorg. Med. Chem. Lett. , 13 629-632, 2004.10

Konno, H.; Hiura, N.; Makabe, H.; Abe, M.; Miyoshi, H.

Multiple Authorship (Including Foreigners)

Synthesis and Mitochondrial Complex I Inhibitoin of Mono- and Non-THF Acetogneins, Proceeding of the 6th Japan/Australia Symposium on Drug Design and Development, 22, 2004.04

Konno, H.; Hiura, H.; Okuno, Y.; Makabe, H.; Hattori, Y.; Miyoshi, H.; Abe, M.; Fujii, N.

Multiple Authorship (Including Foreigners)

Synthesis and mitochondrial complex I inhibition of dihydroxy-cohibin A, non-THF annonaceous acetogenin analogue, BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 14(3) 629-632, 2004.02

Konno, H; Hiura, N; Makabe, H; Abe, M; Miyoshi, H

Single Author

Synthesis of two possible diastereomers of reticulatain-1, TETRAHEDRON LETTERS, 45(5) 973-977, 2004.01

Makabe, H; Miyawaki, A; Takahashi, R; Hattori, Y; Konno, H; Abe, M; Miyoshi, H

Single Author

Efficient Synthesis of Akolactone via Pd-Catalyzed Carbonylation, Biosci. Biotechnol. Biochem., 67(12) 2658-2660, 2003.12

Makabe, H.; Okajima, M.; Konno, H.; Kamo, T.; Hirota, M.

Multiple Authorship (Including Foreigners)

Efficient synthesis of akolactone a <i>via</i> Pd-catalyzed carbonylation, BIOSCIENCE BIOTECHNOLOGY AND BIOCHEMISTRY, 67(12) 2658-2660, 2003.12

Makabe, H; Okajima, M; Konno, H; Kan, T; Hirota, M

Single Author

An Epoxide Ring-Opening Reaction via Hypervalent Silicates Intermediate: Synthesis of Statine, Synthesis, 2161-2164, 2003.11

Konno, H.; Toshiro, E.; Hinoda, N.

Multiple Authorship (Including Foreigners)

An epoxide ring-opening reaction via hypervalent silicate intermediate: Synthesis of statine, SYNTHESIS-STUTTGART, (14) 2161-2164, 2003.10

Konno, H; Toshiro, E; Hinoda, N

Single Author

Structural Revision of Epoxyrollins A and B, Biosynthetic Precursor of Annnonaceous Acetogenins, Biosci. Biotechnol. Biochem., 67(6) 1438-1441, 2003.06

Konno, H.; Makabe, H.

Multiple Authorship (Including Foreigners)

Structural revision of epoxyrollins A and B, biosynthetic precursors of annonaceous acetogenins, BIOSCIENCE BIOTECHNOLOGY AND BIOCHEMISTRY, 67(6) 1438-+, 2003.06

Konno, H; Makabe, H

Single Author

Syntheses of (4S, 5R)- and (4R, 5S)-Muricatacins and (4R, 5S)-aza-muricatacin, Unnatural Analogues of The Annonaceous Acetogenin, Heterocycles, 57(10) 1793-1797, 2002.10

Konno, H.; Hiura, N.; Yanaru, M.

Multiple Authorship (Including Foreigners)

Syntheses of (4<i>R</i>, 5<i>S</i>)- and (4<i>S</i>, 5<i>R</i>)-Muricatacins, and (4<i>S</i>, 5<i>R</i>)-aza-muricatacin, unnatural analogues of the Annonaceous acetogenin, HETEROCYCLES, 57(10) 1793-1797, 2002.10

Konno, H; Hiura, N; Yanaru, M

Single Author

Metal Assisted Stabilization and Probing of Collagenous Triple Helices, J. Am. Chem. Soc. , 124 9388-9289, 2002.09

Koide, T.; Yuguchi, M.; Kawakita, M.; Konno, H.

Multiple Authorship (Including Foreigners)

Metal-assisted stabilization and probing of collagenous triple helices, JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 124(32) 9388-9389, 2002.08

Koide, T; Yuguchi, M; Kawakita, M; Konno, H

Single Author

Preparation of a Synthetic Equivalent of Chiral Methyl 2,5-Dihydroxycyclohexane 1,4-dienecarboxylate, Tetrahedron: Asymmetry, 10 3849-3857, 1999.10

Yoshida, N.; Konno, H.; Kamikubo, T.; Takahashi, M.; Ogasawara, K.

Multiple Authorship (Including Foreigners)

Preparation of a synthetic equivalent of chiral methyl 2,5-dihydroxycyclohexane-1,4-dienecarboxylate, TETRAHEDRON-ASYMMETRY, 10(19) 3849-3857, 1999.09

Yoshida, N; Konno, H; Kamikubo, T; Takahashi, M; Ogasawara, K

Single Author

A Practical Preparation of Versatile Cyclohexenoid Chiral Building Blocks, Synthesis , 1135-1140, 1999.09

Konno, H.; Ogasawara, K.

Multiple Authorship (Including Foreigners)

A practical preparation of versatile cyclohexenoid chiral building blocks, SYNTHESIS-STUTTGART, (7) 1135-1140, 1999.07

Konno, H; Ogasawara, K

Single Author

An enantio- and diastereoselective synthesis of (-)-isoretronecanol and (+)-trachelanthamidine from a <i>meso</i> precursor, HETEROCYCLES, 49 33-37, 1998.12

Konno, H; Kishi, M; Hiroya, K; Ogasawara, K

Single Author

Enantioselective Construction and Utilization of 2-(cyclohex-2-enyl)phenols, Synlett , 1004-1008, 1998.12

Konno, H.; Ogasawara, K.

Multiple Authorship (Including Foreigners)

Enantioselective construction and utilization of 2-(cyclohex-2-enyl)phenols, SYNLETT, (9) 1004-+, 1998.09

Konno, H; Ogasawara, K

Single Author

An Enantio- and Diastereoselective Synthesis of (-)-Isoretronecanol and (+)-Trachelanthamidine from A Meso Precursor, Heterocycles , 49 22-26, 1998.01

Konno, H.; Kishi, M.; Hiroya, K.; Ogasawara, K.

Multiple Authorship (Including Foreigners)

A new tactic for diastereo- and enantiocontrolled synthesis of (-)-malyngolide via catalytic meso-asymmetrization, TETRAHEDRON LETTERS, 38(34) 6023-6026, 1997.08

Konno, H; Hiroya, K; Ogasawara, K

Single Author

A New Tactic for Diastereo- and Enantilcontrolled synthesis of (-)-Malyngolide via Catalytic Meso-Asymmetrization, Tetrahedron Lett. , 38 6023-6026, 1997.01

Konno, H.; Hiroya, K.; Ogasawara, K.

Multiple Authorship (Including Foreigners)

Total Synthesis of (15S, 16R, 19S, 20R, 34S)-Diepomuricanin, Tetrahedron Lett. , 37 5393-5396, 1996.10

Konno, H.; Makabe, H.; Tanaka, A.; Oritani, T.

Multiple Authorship (Including Foreigners)

ynthesis of Two Possible Diastereoisomers of the Epoxy Lactone Proposed for an Annonaceous Acetogenins, Epoxyrollin A, Tetrahedron Lett. , 52 9399-9408, 1996.08

Konno, H.; Makabe, H.; Tanaka, A.; Oritani, T.

Multiple Authorship (Including Foreigners)

Total synthesis of (15S,16R,19S,2OR,34S)-diepomuricanin, TETRAHEDRON LETTERS, 37(30) 5393-5396, 1996.07

Konno, H; Makabe, H; Tanaka, A; Oritani, T

Single Author

Synthetic studies on annonaceous acetogenins .5. Syntheses of two possible diastereoisomers of the epoxy lactone proposed for an annonaceous acetogenin, epoxyrollin A, TETRAHEDRON, 52(28) 9399-9408, 1996.07

Konno, H; Makabe, H; Tanaka, A; Oritani, T

Single Author

Synthesis of Squamostanal-A, Biosci. Biotechnol. Biochem., 60 526-527, 1996.06

Konno, H.; Makabe, H.; Tanaka, A.; Oritani, T.

Multiple Authorship (Including Foreigners)

Synthesis of squamostanal-A, BIOSCIENCE BIOTECHNOLOGY AND BIOCHEMISTRY, 60(3) 526-527, 1996.03

Konno, H; Makabe, H; Tanaka, A; Oritani, T

Single Author

Synthesis of Two Possible Diastereoisomers of the Lactone Proposed for Epoxyrollin A, Biosci. Biotechnol. Biochem., 59 2355-2357, 1995.12

Konno, H.; Makabe, H.; Tanaka, A.; Oritani, T.

Multiple Authorship (Including Foreigners)

Synthetic studies on annonaceous acetogenins .3. Synthesis of two possible diastereoisomers of the epoxy lactone proposed for epoxyrollin A, BIOSCIENCE BIOTECHNOLOGY AND BIOCHEMISTRY, 59(12) 2355-2357, 1995.12

Konno, H; Makabe, H; Tanaka, A; Oritani, T

Single Author