Updated on 2026/04/27

写真a

 
YAMAGUCHI Hiroaki
 
Title
Professor
Date of Birth
1976
Contact information
メールアドレス

Research Areas

  • Life Science / Clinical pharmacy

  • Life Science / Clinical pharmacy

Graduating School

  • Tohoku University, Faculty of Pharmaceutical Science

    1999.03, Graduated

Graduate School

  • Kyoto University, Graduate School, Division of Pharmaceutical Sciences

    Doctor's Course, 2004.03, Completed

External Career

  • Yamagata University, Professor, 2019.04 -

Academic Society Affiliations

  • THE JAPANESE SOCIETY OF CLINICAL PHARMACOLOGY AND THERAPEUTICS

  • JAPANESE SOCIETY FOR BIOMEDICAL MASS SPECTROMETRY

 

Research Career

  • Real-time imaging of carrier-mediated transport, 2007 - 2008

  • Proteomics of bile acid signals, 2008 - 2010

  • Analysis of functional significance of a newly discovered brain-specific transporter, 2008 - 2010

  • Characterization of kidney specific organic anion transporter SLCO4C1, 2011 - 2012

  • Mechanisms of prostanoids release from the cells, 2013.04 - 2016.03

  • Medicinal chemistry studies based on the three-dimensional structural diversity-oriented molecular design of pharmacologically active compounds, 2015.04 - 2020.03

  • Participation of OATP4C1 in the pharmacokinetics of drugs, 2018.04 - 2021.03

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Papers

  • Preparation of TEMPO-Modified Electrodes by Electrochemical Polymerization in Aqueous Solution for Use in Electrochemical Analysis of Pharmaceuticals, ELECTROANALYSIS, 37(10) , 2025.10

    Imahashi, R; Sugiyama, K; Sato, F; Ono, T; Yoshida, K; Kirii, A; Watanabe, K; Yamaguchi, H; Sato, K; Kashiwagi, Y

    Single Author

  • Midnolin gene expression is enhanced by Gq-coupled muscarinic acetylcholine receptor stimulation in SH-SY5Y human neuroblastoma cells, JOURNAL OF PHARMACOLOGICAL SCIENCES, 157(4) 229-232, 2025.04

    Norota, I; Zuiki, Y; Chiba, A; Nagashima, M; Ogura, J; Yamaguchi, H; Ishii, K; Obara, Y

    Single Author

  • Effect of Organic Anion Transporting Polypeptide 1B1 on Plasma Concentration Dynamics of Clozapine in Patients with Treatment-Resistant Schizophrenia, INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 25(23) , 2024.12

    Sato, T; Kawabata, T; Kumondai, M; Hayashi, N; Komatsu, H; Kikuchi, Y; Onoguchi, G; Sato, Y; Nanatani, K; Hiratsuka, M; Maekawa, M; Yamaguchi, H; Abe, T; Tomita, H; Mano, N

    Single Author

  • 臨床決断分析を用いた、遠隔転移を有する大腸癌に対するFOLFIRIベースのファーストライン治療に関する費用対効果分析(Cost-Effectiveness Analysis of FOLFIRI-Based First-Line Regimens for Metastatic Colorectal Cancer Using Clinical Decision Analysis), 癌と化学療法, 51(5) 541-547, 2024.05

    Shida Toshihiro, Ono Yuki, Kobayashi Yuka, Ogura Jiro, Hatakeyama Shiro, Arakawa Ichiro, Inoue Tadao, Yamaguchi Hiroaki

    Single Author

  • The Use of an Antioxidant Enables Accurate Evaluation of the Interaction of Curcumin on Organic Anion-Transporting Polypeptides 4C1 by Preventing Auto-Oxidation, INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 25(2) , 2024.01

    Sato, T; Yagi, A; Yamauchi, M; Kumondai, M; Sato, Y; Kikuchi, M; Maekawa, M; Yamaguchi, H; Abe, T; Mano, N

    Single Author

  • Evaluation of the Efficacy and Limitations of a Simplified Out-of-hospital Prescription Questionnaire-based Protocol through a Questionnaire Survey and Examination of Prescriptions, Iryo Yakugaku (Japanese Journal of Pharmaceutical Health Care and Sciences), 49(12) 423-433, 2023.12

    Ohashi Hiroyo, Kimura Akari, Takahashi Naofumi, Hatakeyama Shiro, Yokomakura Aya, Ogura Jiro, Yamaguchi Hiroaki

    Single Author

  • Architecture for Beyond 5G Services Enabling Cross-Industry Orchestration, IEICE TRANSACTIONS ON COMMUNICATIONS, E106B(12) 1303-1312, 2023.12

    Ishizu, K; Azuma, M; Yamaguchi, H; Kato, A; Hosako, I

    Single Author

  • Cost-Effectiveness Analysis of Cyclin-Dependent Kinase 4/6 Inhibitor Palbociclib for Inoperable or Recurrent Breast Cancer., Gan to kagaku ryoho. Cancer & chemotherapy, 50(8) 895-900, 2023.08

    Toshihiro Shida, Motoko Kaneko, Jiro Ogura, Hiroki Sawada, Shiro Hatakeyama, Ichiro Arakawa, Hiroaki Yamaguchi, Tadao Inoue

    Single Author

  • Acoustic properties for Ga-Sn-Zn liquid metal coupler with low melting point and high acoustic impedance, JAPANESE JOURNAL OF APPLIED PHYSICS, 62(SJ) , 2023.07

    Ohashi, Y; Murakami, R; Yamaguchi, H; Yokota, Y; Yoshikawa, A

    Single Author

  • The effects of prebiotic partially hydrolyzed guar gum on skin hydration: A randomized, open-label, parallel, controlled study in healthy humans, JOURNAL OF FUNCTIONAL FOODS, 103 , 2023.04

    Kapoor, MP; Yamaguchi, H; Ishida, H; Mizutani, Y; Timm, D; Abe, A

    Single Author

  • Glutathione depletion results in S-nitrosylation of protein disulfide isomerase in neuroblastoma cells, LIFE SCIENCES, 316 , 2023.03

    Ono, S; Ogura, J; Sugiura, H; Yamauchi, M; Tanaka, A; Sato, T; Maekawa, M; Yamaguchi, H; Mano, N

    Single Author

  • A hydrolysate of poly-trans -[(2-carboxyethyl)germasesquioxane] (Ge-132) suppresses Cav3.2-dependent pain by sequestering exogenous and endogenous sulfide, REDOX BIOLOGY, 59 , 2023.02

    Sekiguchi, F; Koike, N; Shimada, Y; Sugimoto, K; Masuda, H; Nakamura, T; Yamaguchi, H; Tanabe, G; Marumoto, S; Kasanami, Y; Tsubota, M; Ohkubo, T; Yoshida, S; Kawabata, A

    Single Author

  • Bile Acid-Drug Interaction via Organic Anion-Transporting Polypeptide 4C1 Is a Potential Mechanism of Altered Pharmacokinetics of Renally Excreted Drugs, INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 23(15) , 2022.08

    Yamauchi, M; Sato, T; Otake, A; Kumondai, M; Sato, Y; Kikuchi, M; Maekawa, M; Yamaguchi, H; Abe, T; Mano, N

    Single Author

  • The safety of pranlukast and montelukast during the first trimester of pregnancy: A prospective, two-centered cohort study in Japan, CONGENITAL ANOMALIES, 62(4) 161-168, 2022.07

    Hatakeyama, S; Goto, M; Yamamoto, A; Ogura, J; Watanabe, N; Tsutsumi, S; Yakuwa, N; Yamane, R; Nagase, S; Takahashi, K; Kosaki, R; Murashima, A; Yamaguchi, H

    Single Author

  • The Effectiveness of Antidiabetic Drugs in Treating Dementia: A Peek into Pharmacological and Pharmacokinetic Properties, INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 23(12) , 2022.06

    Ogura, J; Yamaguchi, H

    Single Author

  • KRP-203 Is a Desirable Immunomodulator for Islet Allotransplantation, TRANSPLANTATION, 106(5) 963-972, 2022.05

    Fathi, I; Nishimura, R; Imura, T; Inagaki, A; Kanai, N; Ushiyama, A; Kikuchi, M; Maekawa, M; Yamaguchi, H; Goto, M

    Single Author

  • Glucose-induced oxidative stress leads to in <i>S</i>-nitrosylation of protein disulfide isomerase in neuroblastoma cells, BIOCHIMICA ET BIOPHYSICA ACTA-GENERAL SUBJECTS, 1865(11) , 2021.11

    Ogura, J; Sugiura, H; Tanaka, A; Ono, S; Sato, T; Sato, T; Maekawa, M; Yamaguchi, H; Mano, N

    Single Author

  • Phase II study of trifluridine/tipiracil (TAS-102) therapy in elderly patients with colorectal cancer (T-CORE1401): geriatric assessment tools and plasma drug concentrations as possible predictive biomarkers, CANCER CHEMOTHERAPY AND PHARMACOLOGY, 88(3) 393-402, 2021.09

    Takahashi, M; Sakamoto, Y; Ohori, H; Tsuji, Y; Kuroki, M; Kato, S; Otsuka, K; Komine, K; Takahashi, M; Takahashi, S; Shirota, H; Ouchi, K; Takahashi, Y; Imai, H; Shibata, H; Yoshioka, T; Tanaka, M; Ya...

    Single Author

  • Effect of the Opioid Administration Period before the Initiation of Naldemedine Administration on the Prevalence of Diarrhea(和訳中), 医療薬学, 47(8) 411-417, 2021.08

    Shirata Chinami, Shida Toshihiro, Hatakeyama Shiro, Ogura Jiro, Yamakawa Mayumi, Suzuki Naoki, Yamaguchi Hiroaki

    Single Author

  • Enhancement and evaluation of a prescription audit system for direct oral anticoagulants using a check sheet, JOURNAL OF PHARMACEUTICAL HEALTH CARE AND SCIENCES, 7(1) , 2021.06

    Ishikawa, N; Oshikiri, H; Takasaki, S; Kikuchi, M; Obara, T; Akasaka, K; Matsuura, M; Yamaguchi, H; Mano, N

    Single Author

  • Enhancement and evaluation of a prescription audit system for direct oral anticoagulants using a check sheet(和訳中), Journal of Pharmaceutical Health Care and Sciences, 7 1 of 6-6 of 6, 2021.06

    Ishikawa Naoto, Oshikiri Hanae, Takasaki Shinya, Kikuchi Masafumi, Obara Taku, Akasaka Kazutoshi, Matsuura Masaki, Yamaguchi Hiroaki, Mano Nariyasu

    Single Author

  • Simultaneous analysis of drugs administered to lung-transplanted patients using liquid chromatography-tandem mass spectrometry for therapeutic drug monitoring, BIOMEDICAL CHROMATOGRAPHY, 35(6) , 2021.06

    Takasaki, S; Hirasawa, T; Sato, Y; Maekawa, M; Tsukamoto, T; Kikuchi, M; Ogura, J; Hayakawa, Y; Matsuda, Y; Oishi, H; Sado, T; Noda, M; Okada, Y; Yamaguchi, H; Mano, N

    Single Author

  • Role of OATP4C1 in Renal Handling of Remdesivir and its Nucleoside Analog GS-441524: The First Approved Drug for Patients with COVID-19, JOURNAL OF PHARMACY AND PHARMACEUTICAL SCIENCES, 24 227-236, 2021.05

    Sato, T; Maekawa, M; Mano, N; Abe, T; Yamaguchi, H

    Single Author

  • Development of large size crystal growth technology of oxide eutectic scintillator and a proto-type Talbot-Lau imaging system, JAPANESE JOURNAL OF APPLIED PHYSICS, 60(SB) , 2021.05

    Kamada, K; Yamaguchi, H; Yasui, N; Ohashi, R; Den, T; Kim, KJ; Yoshino, M; Yamaji, A; Kurosawa, S; Shoji, Y; Yokota, Y; Kochurikhin, VV; Yoshikawa, A

    Single Author

  • Azelnidipine treatment reduces the expression of Ca<sub>v</sub>1.2 protein, LIFE SCIENCES, 269 , 2021.03

    Nasu, F; Obara, Y; Okamoto, Y; Yamaguchi, H; Kurakami, K; Norota, I; Ishii, K

    Single Author

  • Clinical Importance of Blood Drug Concentration of Oral Molecular Targeted Drugs for Renal Cell Carcinoma, JOURNAL OF PHARMACY AND PHARMACEUTICAL SCIENCES, 24 127-136, 2021.03

    Takasaki, S; Kawasaki, Y; Kikuchi, M; Ito, A; Yamaguchi, H; Mano, N

    Single Author

  • Knowledge, Attitudes, and Practice of Hospital Pharmacists Regarding Pharmacovigilance and Adverse Drug Reaction Reporting in Japan, HOSPITAL PHARMACY, 56(1) 7-16, 2021.02

    Kobayashi, T; Noda, A; Obara, T; Tsuchiya, M; Akasaka, K; Yoshida, M; Matsuura, M; Sato, M; Murai, Y; Yamaguchi, H; Tsuchiya, F; Kihira, K; Mano, N

    Single Author

  • LARGE-SCALE SYNTHESIS OF THIO-GLUCOSE-CONJUGATED CHLORIN E6 FOR PHOTODYNAMIC THERAPY, HETEROCYCLES, 103(2) 1108-1115, 2021

    Nomoto, A; Yamaguchi, H; Masuda, M; Hyakumura, K; Kodama, S; Osaki, T; Okamoto, Y; Tanaka, M; Kataoka, H; Narumi, A; Yoshimura, T; Yano, S; Ogawa, A

    Single Author

  • Plasma mycophenolic acid concentration and the clinical outcome after lung transplantation, CLINICAL TRANSPLANTATION, 34(12) , 2020.12

    Yabuki, H; Matsuda, Y; Watanabe, T; Eba, S; Hoshi, F; Hirama, T; Oishi, H; Sado, T; Noda, M; Sakurada, A; Kikuchi, M; Yamaguchi, H; Mano, N; Okada, Y

    Single Author

  • Development of a precise quantitative method for monitoring sirolimus in whole blood using LC/ESI-MS/MS, BIOMEDICAL CHROMATOGRAPHY, 34(8) , 2020.08

    Shigeta, K; Kikuchi, M; Tanaka, M; Takasaki, S; Oishi, H; Sado, T; Matsuda, Y; Noda, M; Okada, Y; Mano, N; Yamaguchi, H

    Single Author

  • ATP-Binding Cassette Transporter C4 is a Prostaglandin D2 Exporter in HMC-1 cells, PROSTAGLANDINS LEUKOTRIENES AND ESSENTIAL FATTY ACIDS, 159 , 2020.08

    Tanaka, N; Kawai, J; Hirasawa, N; Mano, N; Yamaguchi, H

    Single Author

  • Selective Chemonucleolysis With Condoliase in Cynomolgus Monkeys, TOXICOLOGIC PATHOLOGY, 48(5) 656-668, 2020.07

    Muramatsu, D; Yamaguchi, H; Minamisawa, Y; Nii, A

    Single Author

  • Stimulatory effect on the transport mediated by organic anion transporting polypeptide 2B1, ASIAN JOURNAL OF PHARMACEUTICAL SCIENCES, 15(2) 181-191, 2020.03

    Ogura, J; Yamaguchi, H; Mano, N

    Single Author

  • Drug Prescriptions for Children With ADHD in Japan: A Study Based on Health Insurance Claims Data Between 2005 and 2015, JOURNAL OF ATTENTION DISORDERS, 24(2) 175-191, 2020.01

    Yoshida, M; Obara, T; Kikuchi, S; Satoh, M; Morikawa, Y; Ooba, N; Yamaguchi, H; Mano, N

    Single Author

  • Comprehensive and semi-quantitative analysis of carboxyl-containing metabolites related to gut microbiota on chronic kidney disease using 2-picolylamine isotopic labeling LC-MS/MS, SCIENTIFIC REPORTS, 9 , 2019.12

    Kanemitsu, Y; Mishima, E; Maekawa, M; Matsumoto, Y; Saigusa, D; Yamaguchi, H; Ogura, J; Tsukamoto, H; Tomioka, Y; Abe, T; Mano, N

    Single Author

  • Investigation of diagnostic performance of five urinary cholesterol metabolites for Niemann-Pick disease type C[S], JOURNAL OF LIPID RESEARCH, 60(12) 2074-2081, 2019.12

    Maekawa, M; Jinnoh, I; Narita, A; Iida, T; Saigusa, D; Iwahori, A; Nittono, H; Okuyama, T; Eto, Y; Ohno, K; Clayton, PT; Yamaguchi, H; Mano, N

    Single Author

  • Risk Factors for Severe Hyponatremia Related to Cisplatin: A Retrospective Case-Control Study, BIOLOGICAL & PHARMACEUTICAL BULLETIN, 42(11) 1891-1897, 2019.11

    Hatakeyama, S; Shida, T; Yamaguchi, H

    Single Author

  • Structural Determination of Lysosphingomyelin-509 and Discovery of Novel Class Lipids from Patients with Niemann-Pick Disease Type C, INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 20(20) , 2019.10

    Maekawa, M; Jinnoh, I; Matsumoto, Y; Narita, A; Mashima, R; Takahashi, H; Iwahori, A; Saigusa, D; Fujii, K; Abe, A; Higaki, K; Yamauchi, S; Ozeki, Y; Shimoda, K; Tomioka, Y; Okuyama, T; Eto, Y; Ohno, ...

    Single Author

  • Estimation of Blood Sirolimus Concentration Based on Tacrolimus Concentration/Dose Normalized by Body Weight Ratio in Lung Transplant Patients, THERAPEUTIC DRUG MONITORING, 41(5) 615-619, 2019.10

    Kikuchi, M; Shigeta, K; Tanaka, M; Takasaki, S; Akiba, M; Oishi, H; Sado, T; Matsuda, Y; Noda, M; Okada, Y; Mano, N; Yamaguchi, H

    Single Author

  • Involvement of H<SUP>+</SUP>-gradient dependent transporter in PGE<sub>2</sub> release from A549 cells, PROSTAGLANDINS LEUKOTRIENES AND ESSENTIAL FATTY ACIDS, 149 30-36, 2019.10

    Tanakaa, N; Yamaguchi, H; Mano, N

    Single Author

  • Organogermanium suppresses cell death due to oxidative stress in normal human dermal fibroblasts, SCIENTIFIC REPORTS, 9 , 2019.09

    Takeda, T; Doiyama, S; Azumi, J; Shimada, Y; Tokuji, Y; Yamaguchi, H; Nagata, K; Sakamoto, N; Aso, H; Nakamura, T

    Single Author

  • Altered bile acid composition and disposition in a mouse model of nonalcoholic steatohepatitis, TOXICOLOGY AND APPLIED PHARMACOLOGY, 379 , 2019.09

    Suga, T; Yamaguchi, H; Ogura, J; Shoji, S; Maekawa, M; Mano, N

    Single Author

  • Limited Sampling Strategy for the Estimation of Mycophenolic Acid and its Acyl Glucuronide Metabolite Area under the Concentration-Time Curve in Japanese Lung Transplant Recipients, JOURNAL OF PHARMACY AND PHARMACEUTICAL SCIENCES, 22 407-417, 2019.08

    Tanaka, S; Kikuchi, M; Takasaki, S; Hirasawa, T; Shigeta, K; Noda, A; Akiba, M; Matsuda, Y; Oishi, H; Sado, T; Noda, M; Okada, Y; Mano, N; Yamaguchi, H

    Single Author

  • Value of global metabolomics in association with diagnosis and clinicopathological factors of renal cell carcinoma, INTERNATIONAL JOURNAL OF CANCER, 145(2) 484-493, 2019.07

    Sato, T; Kawasaki, Y; Maekawa, M; Takasaki, S; Saigusa, D; Ota, H; Shimada, S; Yamashita, S; Mitsuzuka, K; Yamaguchi, H; Ito, A; Kinoshita, K; Koshiba, S; Mano, N; Arai, Y

    Single Author

  • Impact of chronic kidney disease on long-term clinical outcomes of everolimus-eluting stent implantation: A subanalysis of the Tokyo-MD PCI registry, CATHETERIZATION AND CARDIOVASCULAR INTERVENTIONS, 94(1) E9-E16, 2019.07

    Miyazaki, T; Ashikaga, T; Asano, M; Sasaoka, T; Kurihara, K; Yoshikawa, S; Isobe, M; Shimizu, S; Ueshima, D; Yamaguchi, H; Kobayashi, K; Miyazaki, T; Matsumura, A; Sato, Y; Nitta, J; Furubayashi, M; T...

    Single Author

  • Diagnostic performance evaluation of sulfate-conjugated cholesterol metabolites as urinary biomarkers of Niemann-Pick disease type C, CLINICA CHIMICA ACTA, 494 58-63, 2019.07

    Maekawa, M; Narita, A; Jinnoh, I; Iida, T; Marquardt, T; Mengel, E; Eto, Y; Clayton, PT; Yamaguchi, H; Mano, N

    Single Author

  • An immobilized vanadium-binaphthylbishydroxamic acid complex as a reusable catalyst for the asymmetric epoxidation of allylic alcohols, TETRAHEDRON LETTERS, 60(23) 1518-1521, 2019.06

    Noji, M; Kondo, H; Yazaki, C; Yamaguchi, H; Ohkura, S; Takanami, T

    Single Author

  • Analysis of membrane transport mechanisms of endogenous substrates using chromatographic techniques, BIOMEDICAL CHROMATOGRAPHY, 33(6) e4495, 2019.06

    Yamaguchi, H; Mano, N

    Single Author

  • Toward Personalized Cancer Therapy with Oral Molecular-targeted Agents, YAKUGAKU ZASSHI-JOURNAL OF THE PHARMACEUTICAL SOCIETY OF JAPAN, 139(6) 911-915, 2019.06

    Yamaguchi, H; Takasaki, S; Kikuchi, M; Kawasaki, Y; Arai, Y; Mano, N

    Single Author

  • Characterization of conjugated and unconjugated bile acid transport via human organic solute transporter α/β, BIOCHIMICA ET BIOPHYSICA ACTA-BIOMEMBRANES, 1861(5) 1023-1029, 2019.05

    Suga, T; Yamaguchi, H; Ogura, J; Mano, N

    Single Author

  • Fundamental Study of Behaviors of In-Source Collision Induced Dissociation and Shifting the Linear Range of Calibration Curves of Various Drugs and the Metabolites Used for Therapeutic Drug Monitoring., Chromatography, 40(2) 71-78, 2019.05

    Maekawa M, Tsukamoto T, Takasaki S, Kikuchi M, Sato Y, Ogura J, Hayakawa Y, Yamaguchi H, Mano N

    Single Author

  • A Basic Study of Photodynamic Therapy with Glucose-Conjugated Chlorin e6 Using Mammary Carcinoma Xenografts, CANCERS, 11(5) , 2019.05

    Osaki, T; Hibino, S; Yokoe, I; Yamaguchi, H; Nomoto, A; Yano, S; Mikata, Y; Tanaka, M; Kataoka, H; Okamoto, Y

    Single Author

  • Gut microbiome-derived phenyl sulfate contributes to albuminuria in diabetic kidney disease, NATURE COMMUNICATIONS, 10(1) 1835, 2019.04

    Kikuchi, K; Saigusa, D; Kanemitsu, Y; Matsumoto, Y; Thanai, P; Suzuki, N; Mise, K; Yamaguchi, H; Nakamura, T; Asaji, K; Mukawa, C; Tsukamoto, H; Sato, T; Oikawa, Y; Iwasaki, T; Oe, Y; Tsukimi, T; Fuku...

    Single Author

  • Development of a Highly Potent Analogue and a Long-Acting Analogue of Oxytocin for the Treatment of Social Impairment-Like Behaviors, JOURNAL OF MEDICINAL CHEMISTRY, 62(7) 3297-3310, 2019.04

    Ichinose, W; Cherepanov, SM; Shabalova, AA; Yokoyama, S; Yuhi, T; Yamaguchi, H; Watanabe, A; Yamamoto, Y; Okamoto, H; Horike, S; Terakawa, J; Daikoku, T; Watanabe, M; Mano, N; Higashida, H; Shuto, S

    Single Author

  • Long-term relationship between everolimus blood concentration and clinical outcomes in Japanese patients with metastatic renal cell carcinoma: a prospective study., Journal of pharmaceutical health care and sciences, 5 6, 2019

    Takasaki S, Yamaguchi H, Kawasaki Y, Kikuchi M, Tanaka M, Ito A, Mano N

    Single Author

  • Functional characterization of 40 CYP2B6 allelic variants by assessing efavirenz 8-hydroxylation, BIOCHEMICAL PHARMACOLOGY, 156 420-430, 2018.10

    Watanabe, T; Saito, T; Rico, EMG; Hishinuma, E; Kumondai, M; Maekawa, M; Oda, A; Saigusa, D; Saito, S; Yasuda, J; Nagasaki, M; Minegishi, N; Yamamoto, M; Yamaguchi, H; Mano, N; Hirasawa, N; Hiratsuka,...

    Single Author

  • Relationships between sunitinib plasma concentration and clinical outcomes in Japanese patients with metastatic renal cell carcinoma, INTERNATIONAL JOURNAL OF CLINICAL ONCOLOGY, 23(5) 936-943, 2018.10

    Takasaki, S; Kawasaki, Y; Kikuchi, M; Tanaka, M; Suzuka, M; Noda, A; Sato, Y; Yamashita, S; Mitsuzuka, K; Saito, H; Ito, A; Yamaguchi, H; Arai, Y; Mano, N

    Single Author

  • Functional Characterization of 21 Allelic Variants of Dihydropyrimidine Dehydrogenase Identified in 1070 Japanese Individuals, DRUG METABOLISM AND DISPOSITION, 46(8) 1083-1090, 2018.08

    Hishinuma, E; Narita, Y; Saito, S; Maekawa, M; Akai, F; Nakanishi, Y; Yasuda, J; Nagasaki, M; Yamamoto, M; Yamaguchi, H; Mano, N; Hirasawa, N; Hiratsuka, M

    Single Author

  • Optimization of Dopants and Scintillation Fibers' Diameter of GdAlO<sub>3</sub>/α-Al<sub>2</sub>O<sub>3</sub> Eutectic for High-Resolution X-Ray Imaging, IEEE TRANSACTIONS ON NUCLEAR SCIENCE, 65(8) 2036-2040, 2018.08

    Kamada, K; Yasui, N; Ohashi, Y; Den, T; Yamaguchi, H; Yamaji, A; Shoji, Y; Yoshisno, M; JinKim, K; Kurosawa, S; Ohashi, Y; Yokota, Y; Yoshikawa, A

    Single Author

  • Simultaneous analysis of oral anticancer drugs for renal cell carcinoma in human plasma using liquid chromatography/electrospray ionization tandem mass spectrometry, BIOMEDICAL CHROMATOGRAPHY, 32(6) e4184, 2018.06

    Takasaki, S; Tanaka, M; Kikuchi, M; Maekawa, M; Kawasaki, Y; Ito, A; Arai, Y; Yamaguchi, H; Mano, N

    Single Author

  • 肺移植患者における個別化薬物療法, 臨床薬理の進歩, (39) 104-116, 2018.06

    山口 浩明, 菊地 正史, 田中 雅樹, 高崎 新也, 野田 あおい, 重田 健介, 白木 美香, 高木 秀侑, 松田 安史, 野田 雅史, 岡田 克典, 眞野 成康

    Single Author

  • Possible predictive value of G8 score and the drug concentrations for efficacy and toxicity of trifluridine/tipiracil for elderly patients with advanced colorectal cancer: A multicenter, phase II study (T-CORE1401)., JOURNAL OF CLINICAL ONCOLOGY, 36(15) , 2018.05

    Takahashi, M; Gamoh, M; Ohori, H; Sakamoto, Y; Tsuji, Y; Kuroki, M; Takahashi, M; Yaegashi, H; Yamaguchi, H; Yamaguchi, T; Shimodaira, H; Yoshioka, T; Ishioka, C

    Single Author

  • Impact of clinical factors and UGT1A9 and CYP2B6 genotype on inter-individual differences in propofol pharmacokinetics, JOURNAL OF ANESTHESIA, 32(2) 236-243, 2018.04

    Kanaya, A; Sato, T; Fuse, N; Yamaguchi, H; Mano, N; Yamauchi, M

    Single Author

  • Mg, Ce co-doped Lu<sub>2</sub>Gd<sub>1</sub>(Ga,Al)<sub>5</sub>O<sub>12</sub> by micro-pulling down method and their luminescence properties, JAPANESE JOURNAL OF APPLIED PHYSICS, 57(4) , 2018.04

    Kamada, K; Yamaguchi, H; Yoshino, M; Kurosawa, S; Shoji, Y; Yokota, Y; Ohashi, Y; Pejchal, J; Nikl, M; Yoshikawa, A

    Single Author

  • Excellent antitumor effects for gastrointestinal cancers using photodynamic therapy with a novel glucose conjugated chlorin e6, BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 496(4) 1204-1209, 2018.02

    Nishie, H; Kataoka, H; Yano, S; Yamaguchi, H; Nomoto, A; Tanaka, M; Kato, A; Shimura, T; Mizoshita, T; Kubota, E; Tanida, S; Joh, T

    Single Author

  • Functional characterization of 9 CYP2A13 allelic variants by assessment of nicotine <i>C</i>-oxidation and coumarin 7-hydroxylation, DRUG METABOLISM AND PHARMACOKINETICS, 33(1) 82-89, 2018.02

    Kumondai, M; Hosono, H; Maekawa, M; Yamaguchi, H; Mano, N; Oda, A; Hirasawa, N; Hiratsuka, M

    Single Author

  • Comparison of PETINIA and LC-MS/MS for determining plasma mycophenolic acid concentrations in Japanese lung transplant recipients., Journal of pharmaceutical health care and sciences, 4 7, 2018

    Kikuchi M, Tanaka M, Takasaki S, Takahashi A, Akiba M, Matsuda Y, Noda M, Hisamichi K, Yamaguchi H, Okada Y, Mano N

    Single Author

  • Interactions of crizotinib and gefitinib with organic anion-transporting polypeptides (OATP)1B1, OATP1B3 and OATP2B1: gefitinib shows contradictory interaction with OATP1B3, XENOBIOTICA, 48(1) 73-78, 2018

    Sato, T; Ito, H; Hirata, A; Abe, T; Mano, N; Yamaguchi, H

    Single Author

  • Development of a Liquid Chromatography-Tandem Mass Spectrometric Method for Quantification of Mycophenolic Acid and Its Glucuronides in Dried Blood Spot Samples, THERAPEUTIC DRUG MONITORING, 39(6) 648-653, 2017.12

    Iboshi, H; Yamaguchi, H; Suzuki, H; Kikuchi, M; Tanaka, M; Takasaki, S; Takahashi, A; Maekawa, M; Shimada, M; Matsuda, Y; Okada, Y; Mano, N

    Single Author

  • Functional characterization of 21 allelic variants of dihydropyrimidinase, BIOCHEMICAL PHARMACOLOGY, 143 118-128, 2017.11

    Hishinuma, E; Akai, F; Narita, Y; Maekawa, M; Yamaguchi, H; Mano, N; Oda, A; Hirasawa, N; Hiratsuka, M

    Single Author

  • Potential Drug Interactions Mediated by Renal Organic Anion Transporter OATP4C1, JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 362(2) 271-277, 2017.08

    Sato, T; Mishima, E; Mano, N; Abe, T; Yamaguchi, H

    Single Author

  • Mitochonic Acid 5 (MA-5) Facilitates ATP Synthase Oligomerization and Cell Survival in Various Mitochondrial Diseases, EBIOMEDICINE, 20 27-38, 2017.06

    Matsuhashi, T; Sato, T; Kanno, S; Suzuki, T; Matsuo, A; Oba, Y; Kikusato, M; Ogasawara, E; Kudo, T; Suzuki, K; Ohara, O; Shimbo, H; Nanto, F; Yamaguchi, H; Saigusa, D; Mukaiyama, Y; Watabe, A; Kikuchi...

    Single Author

  • Analytical Technologies Used in the Medical Front, BUNSEKI KAGAKU, 66(6) 413-419, 2017.06

    Maekawa, M; Yamaguchi, H; Mano, N

    Single Author

  • Matrix effect-corrected liquid chromatography/tandem mass-spectrometric method for determining acylcarnitines in human urine, CLINICA CHIMICA ACTA, 468 187-194, 2017.05

    Abe, K; Suzuki, H; Maekawa, M; Shimada, M; Yamaguchi, H; Mano, N

    Single Author

  • Activation of the Hypoxia Inducible Factor 1α Subunit Pathway in Steatotic Liver Contributes to Formation of Cholesterol Gallstones, GASTROENTEROLOGY, 152(6) 1521-+, 2017.05

    Asai, Y; Yamada, T; Tsukita, S; Takahashi, K; Maekawa, M; Honma, M; Ikeda, M; Murakami, K; Munakata, Y; Shirai, Y; Kodama, S; Sugisawa, T; Chiba, Y; Kondo, Y; Kaneko, K; Uno, K; Sawada, S; Imai, J; Na...

    Single Author

  • Comparison of Concentration Methods for Low-level Radiocesium in Fresh Water, BUNSEKI KAGAKU, 66(4) 299-307, 2017.04

    Yasutaka, T; Shin, M; Onda, Y; Shinano, T; Hayashi, S; Tsukada, H; Aono, T; Iijima, K; Eguchi, S; Ohno, K; Yoshida, Y; Kamihigashi, H; Kitamura, K; Kubota, T; Nogawa, N; Yoshikawa, N; Yamaguchi, H; Su...

    Single Author

  • Functional Characterization of 34 CYP2A6 Allelic Variants by Assessment of Nicotine <i>C</i>-Oxidation and Coumarin 7-Hydroxylation Activities, DRUG METABOLISM AND DISPOSITION, 45(3) 279-285, 2017.03

    Hosono, H; Kumondai, M; Maekawa, M; Yamaguchi, H; Mano, N; Oda, A; Hirasawa, N; Hiratsuka, M

    Single Author

  • Effects of Mg-codoping on luminescence and scintillation properties of Ce doped Lu<sub>3</sub>(Ga,Al)<sub>5</sub>O<sub>12</sub> single crystals, OPTICAL MATERIALS, 65 60-65, 2017.03

    Yamaguchi, H; Kamada, K; Pejchal, J; Kurosawa, S; Shoji, Y; Yokota, Y; Ohashi, Y; Yoshikawa, A

    Single Author

  • Severe toxicity induced by accumulation of active sunitinib metabolite in a Japanese patient with renal cell carcinoma: a case report., Journal of medical case reports, 11(1) 28, 2017.02

    Takasaki S, Kikuchi M, Kawasaki Y, Ito A, Arai Y, Yamaguchi H, Mano N

    Single Author

  • Preference of Conjugated Bile Acids over Unconjugated Bile Acids as Substrates for OATP1B1 and OATP1B3, PLOS ONE, 12(1) e0169719, 2017.01

    Suga, T; Yamaguchi, H; Sato, T; Maekawa, M; Goto, J; Mano, N

    Single Author

  • [A Case of Renal Cell Carcinoma with High Everolimus Blood Concentrations and Hyperglycemia Due to Everolimus-Induced Hepatic Dysfunction]., Gan to kagaku ryoho. Cancer & chemotherapy, 44(1) 87-89, 2017.01

    Takasaki S, Kikuchi M, Kawasaki Y, Ito A, Arai Y, Yamaguchi H, Mano N

    Single Author

  • A simultaneous determination method for 5-fluorouracil and its metabolites in human plasma with linear range adjusted by in-source collision-induced dissociation using hydrophilic interaction liquid chromatography-electrospray ionization-tandem mass spectrometry, BIOMEDICAL CHROMATOGRAPHY, 30(11) 1882-1886, 2016.11

    Ishii, H; Shimada, M; Yamaguchi, H; Mano, N

    Single Author

  • Co-doping effects on luminescence and scintillation properties of Ce doped (Lu,Gd)<sub>3</sub>(Ga,Al)<sub>5</sub>O<sub>12</sub> scintillator, OPTICAL MATERIALS, 61 129-133, 2016.11

    Yamaguchi, H; Kamada, K; Kurosawa, S; Pejchal, J; Shoji, Y; Yokota, Y; Ohashi, Y; Yoshikawa, A

    Single Author

  • Mitochonic Acid 5 Binds Mitochondria and Ameliorates Renal Tubular and Cardiac Myocyte Damage, JOURNAL OF THE AMERICAN SOCIETY OF NEPHROLOGY, 27(7) 1925-1932, 2016.07

    Suzuki, T; Yamaguchi, H; Kikusato, M; Hashizume, O; Nagatoishi, S; Matsuo, A; Sato, T; Kudo, T; Matsuhashi, T; Murayanna, K; Ohba, Y; Watanabe, S; Kanno, S; Minaki, D; Saigusa, D; Shinbo, H; Mori, N; ...

    Single Author

  • Shifting the Linear Range in Electrospray Ionization by In-Source Collision-Induced Dissociation, CHEMICAL & PHARMACEUTICAL BULLETIN, 64(4) 356-359, 2016.04

    Ishii, H; Yamaguchi, H; Mano, N

    Single Author

  • Trough blood levels of sunitinib for Asian (Japanese) patients with metastatic renal cell carcinoma and therapeutic drug monitoring., JOURNAL OF CLINICAL ONCOLOGY, 34(2) , 2016.01

    Kawasaki, Y; Takasaki, S; Ito, A; Mitsuzuka, K; Yamashita, S; Kawamorita, N; Izumi, H; Adachi, H; Kaiho, Y; Tanaka, M; Kikuchi, M; Yamaguchi, H; Mano, N; Arai, Y

    Single Author

  • Identification of Two Sulfated Cholesterol Metabolites Found in the Urine of a Patient with Niemann-Pick Disease Type C as Novel Candidate Diagnostic Markers., Mass spectrometry (Tokyo, Japan), 5(2) S0053, 2016

    Maekawa M, Omura K, Sekiguchi S, Iida T, Saigusa D, Yamaguchi H, Mano N

    Single Author

  • Special Issue on Intelligent Autonomous Systems, ROBOTICS AND AUTONOMOUS SYSTEMS, 74 297-298, 2015.12

    Menegatti, E; Berns, K; Michael, N; Yamaguchi, H

    Single Author

  • ORGANIC ANION TRANSPORTING POLYPEPTIDES 1B1 AND 1B3 PLAY AN IMPORTANT ROLE IN UREMIC TOXIN HANDLING AND DRUG-UREMIC TOXIN INTERACTIONS IN THE LIVER, DRUG METABOLISM REVIEWS, 47 264-265, 2015.11

    Sato, T; Yamaguchi, H; Kogawa, T; Abe, T; Mano, N

    Single Author

  • IDENTIFICATION OF THE OATP1B3-SPECIFIC COMPOUND LST-02, DRUG METABOLISM REVIEWS, 47 255-256, 2015.11

    Yamaguchi, H; Abe, T; Mano, N

    Single Author

  • Profiles of Immune Cells and Reproduction of Immune-mediated Drug-induced Liver Injury, AMERICAN JOURNAL OF GASTROENTEROLOGY, 110 S871, 2015.10

    Fujisaka, Y; Kondo, Y; Sasaki, T; Kogure, T; Inoue, J; Nakagome, Y; Wakui, Y; Iwata, T; Morosawa, T; Umetsu, T; Suzuki, H; Yamaguchi, H; Mano, N; Nagata, K; Shimosegawa, T

    Single Author

  • Reactive oxygen species derived from xanthine oxidase interrupt dimerization of breast cancer resistance protein, resulting in suppression of uric acid excretion to the intestinal lumen, BIOCHEMICAL PHARMACOLOGY, 97(1) 89-98, 2015.09

    Ogura, J; Kuwayama, K; Sasaki, S; Kaneko, C; Koizumi, T; Yabe, K; Tsujimoto, T; Takeno, R; Takaya, A; Kobayashi, M; Yamaguchi, H; Iseki, K

    Single Author

  • Successful Colistin Treatment of Multidrug-Resistant <i>Pseudomonas aeruginosa</i> Infection Using a Rapid Method for Determination of Colistin in Plasma: Usefulness of Therapeutic Drug Monitoring, BIOLOGICAL & PHARMACEUTICAL BULLETIN, 38(9) 1430-1433, 2015.09

    Yamada, T; Ishiguro, N; Oku, K; Higuchi, I; Nakagawa, I; Noguchi, A; Yasuda, S; Fukumoto, T; Iwasaki, S; Akizawa, K; Furugen, A; Yamaguchi, H; Iseki, K

    Single Author

  • Focused metabolomics using liquid chromatography/electrospray ionization tandem mass spectrometry for analysis of urinary conjugated cholesterol metabolites from patients with Niemann-Pick disease type C and 3-hydroxysteroid dehydrogenase deficiency, ANNALS OF CLINICAL BIOCHEMISTRY, 52(5) 576-587, 2015.09

    Maekawa, M; Shimada, M; Ohno, K; Togawa, M; Nittono, H; Iida, T; Hofmann, AF; Goto, J; Yamaguchi, H; Mano, N

    Single Author

  • Mitochonic Acid 5 (MA-5), a Derivative of the Plant Hormone Indole-3-Acetic Acid, Improves Survival of Fibroblasts from Patients with Mitochondrial Diseases, TOHOKU JOURNAL OF EXPERIMENTAL MEDICINE, 236(3) 225-232, 2015.07

    Suzuki, T; Yamaguchi, H; Kikusato, M; Matsuhashi, T; Matsuo, A; Sato, T; Oba, Y; Watanabe, S; Minaki, D; Saigusa, D; Shimbo, H; Mori, N; Mishima, E; Shima, H; Akiyama, Y; Takeuchi, Y; Yuri, A; Kikuchi...

    Single Author

  • Simultaneous quantification of leukotrienes and hydroxyeicosatetraenoic acids in cell culture medium using liquid chromatography/tandem mass spectrometry, BIOMEDICAL CHROMATOGRAPHY, 29(7) 1084-1093, 2015.07

    Furugen, A; Yamaguchi, H; Mano, N

    Single Author

  • Involvement of Histidine Residue His382 in pH Regulation of MCT4 Activity, PLOS ONE, 10(4) e0122738, 2015.04

    Sasaki, S; Kobayashi, M; Futagi, Y; Ogura, J; Yamaguchi, H; Iseki, K

    Single Author

  • Determination of ω-6 and ω-3 PUFA metabolites in human urine samples using UPLC/MS/MS (vol 407, pg 1625, 2015), ANALYTICAL AND BIOANALYTICAL CHEMISTRY, 407(10) 2939-2940, 2015.04

    Sasaki, A; Fukuda, H; Shiida, N; Tanaka, N; Furugen, A; Ogura, J; Shuto, S; Mano, N; Yamaguchi, H

    Single Author

  • A Novel Extraction Method Based on a Reversible Chemical Conversion for the LC/MS/MS Analysis of the Stable Organic Germanium Compound Ge-132, ANALYTICAL CHEMISTRY, 87(4) 2042-2047, 2015.02

    Yamaguchi, H; Shimada, Y; Takeda, T; Nakamura, T; Mano, N

    Single Author

  • Determination of ω-6 and ω-3 PUFA metabolites in human urine samples using UPLC/MS/MS, ANALYTICAL AND BIOANALYTICAL CHEMISTRY, 407(6) 1625-1639, 2015.02

    Sasaki, A; Fukuda, H; Shiida, N; Tanaka, N; Furugen, A; Ogura, J; Shuto, S; Mano, N; Yamaguchi, H

    Single Author

  • Control of two manipulation points of a cooperative transportation system with two car-like vehicles following parametric curve paths, ROBOTICS AND AUTONOMOUS SYSTEMS, 63 165-178, 2015.01

    Yamaguchi, H; Nishijima, A; Kawakami, A

    Single Author

  • Quantification of intracellular and extracellular digoxin and ouabain by liquid chromatography/electrospray ionization tandem mass spectrometry, JOURNAL OF CHROMATOGRAPHY B-ANALYTICAL TECHNOLOGIES IN THE BIOMEDICAL AND LIFE SCIENCES, 972 73-80, 2014.12

    Yamaguchi, H; Miyamori, K; Sato, T; Ogura, J; Kobayashi, M; Yamada, T; Mano, N; Iseki, K

    Single Author

  • Transport of Eicosapentaenoic Acid-Derived PGE<sub>3</sub>, PGF<sub>3α</sub>, and TXB<sub>3</sub> by ABCC4, PLOS ONE, 9(10) , 2014.10

    Tanaka, N; Yamaguchi, H; Mano, N

    Single Author

  • Quantification of intracellular and extracellular eicosapentaenoic acid-derived 3-series prostanoids by liquid chromatography/electrospray ionization tandem mass spectrometry, PROSTAGLANDINS LEUKOTRIENES AND ESSENTIAL FATTY ACIDS, 91(3) 61-71, 2014.09

    Tanaka, N; Yamaguchi, H; Furugen, A; Ogura, J; Kobayashi, M; Yamada, T; Mano, N; Iseki, K

    Single Author

  • Quercetin-3-rhamnoglucoside (rutin) stimulates transport of organic anion compounds mediated by organic anion transporting polypeptide 2B1, BIOPHARMACEUTICS & DRUG DISPOSITION, 35(3) 173-182, 2014.04

    Ogura, J; Koizumi, T; Segawa, M; Yabe, K; Kuwayama, K; Sasaki, S; Kaneko, C; Tsujimoto, T; Kobayashi, M; Yamaguchi, H; Iseki, K

    Single Author

  • Immunoprotective Effect of Epigallocatechin-3-gallate on Oral Anticancer Drug-Induced α-Defensin Reduction in Caco-2 Cells, BIOLOGICAL & PHARMACEUTICAL BULLETIN, 37(3) 490-492, 2014.03

    Takahashi, N; Kobayashi, M; Ogura, J; Yamaguchi, H; Satoh, T; Watanabe, K; Iseki, K

    Single Author

  • ACTIVATION OF XANTHINE OXIDASE SUPPRESSES DISULFIDE BOND FORMATION OF BREAST CANCER RESISTANCE PROTEIN IN CACO-2 CELLS, DRUG METABOLISM REVIEWS, 45 265, 2014.01

    Ogura, J; Sasaki, S; Kuwayama, K; Kaneko, C; Koizumi, T; Yabe, K; Yamaguchi, H; Iseki, K

    Single Author

  • Intestinal P-glycoprotein expression is multimodally regulated by intestinal ischemia-reperfusion., J Pharm Pharm Sci, 17(2) 266-276, 2014

    Terada, Yusuke Ogura, Jiro Tsujimoto, Takashi Kuwayama, Kaori Koizumi, Takahiro Sasaki, Shunichi Maruyama, Hajime Kobayashi, Masaki Yamaguchi, Hiroaki Iseki, Ken

    Single Author

  • Organic Anion Transporting Polypeptides 1B1 and 1B3 Play an Important Role in Uremic Toxin Handling and Drug-Uremic Toxin Interactions in the Liver, JOURNAL OF PHARMACY AND PHARMACEUTICAL SCIENCES, 17(4) 475-484, 2014

    Sato, T; Yamaguchi, H; Kogawa, T; Abe, T; Mano, N

    Single Author

  • Alteration of pharmacokinetics of grepafloxacin in type 2 diabetic rats., J Pharm Pharm Sci, 17(1) 25-33, 2014

    Watanabe, Meguho Kobayashi, Masaki Ogura, Jiro Takahashi, Natsuko Yamaguchi, Hiroaki Iseki, Ken

    Single Author

  • Intestinal P-glycoprotein Expression is Multimodally Regulated by Intestinal Ischemia-Reperfusion, JOURNAL OF PHARMACY AND PHARMACEUTICAL SCIENCES, 17(2) 266-276, 2014

    Terada, Y; Ogura, J; Tsujimoto, T; Kuwayama, K; Koizumi, T; Sasaki, S; Maruyama, H; Kobayashi, M; Yamaguchi, H; Iseki, K

    Single Author

  • Alteration of Pharmacokinetics of Grepafloxacin in Type 2 Diabetic Rats, JOURNAL OF PHARMACY AND PHARMACEUTICAL SCIENCES, 17(1) 25-33, 2014

    Watanabe, M; Kobayashi, M; Ogura, J; Takahashi, N; Yamaguchi, H; Iseki, K

    Single Author

  • Effect of oxidative stress on expression and function of human and rat organic anion transporting polypeptides in the liver., Int J Pharm, 458(2) 262-271, 2013.12

    Tsujimoto, Takashi Ogura, Jiro Kuwayama, Kaori Koizumi, Takahiro Sasaki, Shunichi Terada, Yusuke Kobayashi, Masaki Yamaguchi, Hiroaki Iseki, Ken

    Single Author

  • Megalin Contributes to Kidney Accumulation and Nephrotoxicity of Colistin, ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 57(12) 6319-6324, 2013.12

    Suzuki, T; Yamaguchi, H; Ogura, J; Kobayashi, M; Yamada, T; Iseki, K

    Single Author

  • Effect of oxidative stress on expression and function of human and rat organic anion transporting polypeptides in the liver., Int J Pharm, 2013.10

    Tsujimoto, Takashi Ogura, Jiro Kuwayama, Kaori Koizumi, Takahiro Sasaki, Shunichi Terada, Yusuke Kobayashi, Masaki Yamaguchi, Hiroaki Iseki, Ken

    Single Author

  • Contribution of multidrug resistance-associated proteins (MRPs) to the release of prostanoids from A549 cells, PROSTAGLANDINS & OTHER LIPID MEDIATORS, 106 37-44, 2013.10

    Furugen, A; Yamaguchi, H; Tanaka, N; Shiida, N; Ogura, J; Kobayashi, M; Iseki, K

    Single Author

  • LC/ESI-MS/MS analysis of urinary 3β-sulfooxy-7β-<i>N</i>-acetylglucosaminyl-5-cholen-24-oic acid and its amides: New biomarkers for the detection of Niemann-Pick type C disease, STEROIDS, 78(10) 967-972, 2013.10

    Maekawa, M; Misawa, Y; Sotoura, A; Yamaguchi, H; Togawa, M; Ohno, K; Nittono, H; Kakiyama, G; Iida, T; Hofmann, AF; Goto, J; Shimada, M; Mano, N

    Single Author

  • Regulation of the Expression and Activity of Glucose and Lactic Acid Metabolism-Related Genes by Protein Kinase C in Skeletal Muscle Cells, BIOLOGICAL & PHARMACEUTICAL BULLETIN, 36(9) 1435-1439, 2013.09

    Otake, S; Kobayashi, M; Narumi, K; Sasaki, S; Kikutani, Y; Furugen, A; Watanabe, M; Takahashi, N; Ogura, J; Yamaguchi, H; Iseki, K

    Single Author

  • Regulation of multidrug resistance protein 2 (MRP2, ABCC2) expression by statins: Involvement of SREBP-mediated gene regulation, INTERNATIONAL JOURNAL OF PHARMACEUTICS, 452(1-2) 36-41, 2013.08

    Kobayashi, M; Gouda, K; Chisaki, I; Asada, K; Ogura, J; Takahashi, N; Konishi, T; Koshida, Y; Sasaki, S; Yamaguchi, H; Iseki, K

    Single Author

  • Crucial Residue Involved in L-Lactate Recognition by Human Monocarboxylate Transporter 4 (hMCT4), PLOS ONE, 8(7) e67690, 2013.07

    Sasaki, S; Kobayashi, M; Futagi, Y; Ogura, J; Yamaguchi, H; Takahashi, N; Iseki, K

    Single Author

  • Rapid Stimulating Effect of the Antiarrhythmic Agent Amiodarone on Absorption of Organic Anion Compounds, DRUG METABOLISM AND PHARMACOKINETICS, 28(3) 178-186, 2013.06

    Segawa, M; Ogura, J; Seki, S; Itagaki, S; Takahashi, N; Kobayashi, M; Hirano, T; Yamaguchi, H; Iseki, K

    Single Author

  • Chondroitinase injection improves keloid pathology by reorganizing the extracellular matrix with regenerated elastic fibers, JOURNAL OF DERMATOLOGY, 40(5) 380-383, 2013.05

    Ishiko, T; Naitoh, M; Kubota, H; Yamawaki, S; Ikeda, M; Yoshikawa, K; Fujita, H; Yamaguchi, H; Kurahashi, Y; Suzuki, S

    Single Author

  • Quantitative determination of paclitaxel and its metabolites, 6α-hydroxypaclitaxel and p-3′-hydroxypaclitaxel, in human plasma using column-switching liquid chromatography/tandem mass spectrometry, BIOMEDICAL CHROMATOGRAPHY, 27(4) 539-544, 2013.04

    Yamaguchi, H; Fujikawa, A; Ito, H; Tanaka, N; Furugen, A; Miyamori, K; Takahashi, N; Ogura, J; Kobayashi, M; Yamada, T; Mano, N; Iseki, K

    Single Author

  • Renal uptake of substrates for organic anion transporters Oat1 and Oat3 and organic cation transporters Oct1 and Oct2 is altered in rats with adenine-induced chronic renal failure, JOURNAL OF PHARMACEUTICAL SCIENCES, 102(3) 1086-1094, 2013.03

    Komazawa, H; Yamaguchi, H; Hidaka, K; Ogura, J; Kobayashi, M; Iseki, K

    Single Author

  • Quantification of intact carboplatin in human plasma ultrafitrates using hydrophilic interaction liquid chromatography-tandem mass spectrometry and its application to a pharmacokinetic study, JOURNAL OF CHROMATOGRAPHY B-ANALYTICAL TECHNOLOGIES IN THE BIOMEDICAL AND LIFE SCIENCES, 917 18-23, 2013.02

    Ito, H; Yamaguchi, H; Fujikawa, A; Shiida, N; Tanaka, N; Ogura, J; Kobayashi, M; Yamada, T; Mano, N; Iseki, K

    Single Author

  • Intestinal ischemia-reperfusion suppresses biliary excretion of hepatic organic anion transporting polypeptides substrate., J Pharm Pharm Sci, 16(5) 722-731, 2013

    Maruyama, Hajime Ogura, Jiro Fujikawa, Asuka Terada, Yusuke Tsujimoto, Takashi Koizumi, Takahiro Kuwayama, Kaori Kobayashi, Masaki Yamaguchi, Hiroaki Iseki, Ken

    Single Author

  • Regulation of the expression and activity of glucose and lactic acid metabolism-related genes by protein kinase C in skeletal muscle cells., Biol Pharm Bull, 36(9) 1435-1439, 2013

    Otake, Sho Kobayashi, Masaki Narumi, Katsuya Sasaki, Shotaro Kikutani, Yurika Furugen, Ayako Watanabe, Meguho Takahashi, Natsuko Ogura, Jiro Yamaguchi, Hiroaki Iseki, Ken

    Single Author

  • Intestinal Ischemia-Reperfusion Suppresses Biliary Excretion of Hepatic Organic Anion Transporting Polypeptides Substrate, JOURNAL OF PHARMACY AND PHARMACEUTICAL SCIENCES, 16(5) 722-731, 2013

    Maruyama, H; Ogura, J; Fujikawa, A; Terada, Y; Tsujimoto, T; Koizumi, T; Kuwayama, K; Kobayashi, M; Yamaguchi, H; Iseki, K

    Single Author

  • A full validated hydrophilic interaction liquid chromatography-tandem mass spectrometric method for the quantification of oxaliplatin in human plasma ultrafiltrates, JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 71 99-103, 2012.12

    Ito, H; Yamaguchi, H; Fujikawa, A; Tanaka, N; Furugen, A; Miyamori, K; Takahashi, N; Ogura, J; Kobayashi, M; Yamada, T; Mano, N; Iseki, K

    Single Author

  • Usefulness of Low Dose Pimobendan in Addition to Conventional Therapy in Patients with Severe Congestive Heart Failure, JOURNAL OF CARDIAC FAILURE, 18(10) S181, 2012.10

    Okazaki, H; Itoh, S; Tanii, H; Yamaguchi, H; Sakurada, H; Hiraoka, M

    Single Author

  • Repair of silorane-based dental composites: Influence of surface treatments, DENTAL MATERIALS, 28(8) 894-902, 2012.08

    Hamano, N; Chiang, YC; Nyamaa, I; Yamaguchi, H; Ino, S; Hickel, R; Kunzelmann, KH

    Single Author

  • Simultaneous quantitation of sphingoid bases and their phosphates in biological samples by liquid chromatography/electrospray ionization tandem mass spectrometry, ANALYTICAL AND BIOANALYTICAL CHEMISTRY, 403(7) 1897-1905, 2012.06

    Saigusa, D; Shiba, K; Inoue, A; Hama, K; Okutani, M; Iida, N; Saito, M; Suzuki, K; Kaneko, T; Suzuki, N; Yamaguchi, H; Mano, N; Goto, J; Hishinuma, T; Aoki, J; Tomioka, Y

    Single Author

  • Regulation of human monocarboxylate transporter 4 in skeletal muscle cells: The role of protein kinase C (PKC), INTERNATIONAL JOURNAL OF PHARMACEUTICS, 428(1-2) 25-32, 2012.05

    Narumi, K; Kobayashi, M; Otake, S; Furugen, A; Takahashi, N; Ogura, J; Itagaki, S; Hirano, T; Yamaguchi, H; Iseki, K

    Single Author

  • Effects of Acidification and Alkalinization Agent on Statins-induced Muscle Toxicity, YAKUGAKU ZASSHI-JOURNAL OF THE PHARMACEUTICAL SOCIETY OF JAPAN, 132(5) 609-615, 2012.05

    Kobayashi, M; Hidaka, K; Chisaki, I; Takahashi, N; Ogura, J; Itagaki, S; Hirano, T; Yamaguchi, H; Iseki, K

    Single Author

  • Examination of bond strength and mechanical properties of Y-TZP zirconia ceramics with different surface modifications, DENTAL MATERIALS JOURNAL, 31(3) 472-480, 2012.05

    Yamaguchi, H; Ino, S; Hamano, N; Okada, S; Teranaka, T

    Single Author

  • A rapid and sensitive LC/ESI-MS/MS method for quantitative analysis of docetaxel in human plasma and its application to a pharmacokinetic study, JOURNAL OF CHROMATOGRAPHY B-ANALYTICAL TECHNOLOGIES IN THE BIOMEDICAL AND LIFE SCIENCES, 893 157-161, 2012.04

    Yamaguchi, H; Fujikawa, A; Ito, H; Tanak, N; Furugen, A; Miyamori, K; Takahashi, N; Ogura, J; Kobayashi, M; Yamada, T; Mano, N; Iseki, K

    Single Author

  • The decrease in farnesoid X receptor, pregnane X receptor and constitutive androstane receptor in the liver after intestinal ischemia-reperfusion., J Pharm Pharm Sci, 15(5) 616-631, 2012

    Ogura, Jiro Terada, Yusuke Tsujimoto, Takashi Koizumi, Takahiro Kuwayama, Kaori Maruyama, Hajime Fujikawa, Asuka Takaya, Atsushi Kobayashi, Masaki Itagaki, Shirou Takahashi, Natsuko Hirano, Takeshi Ya...

    Single Author

  • Intestinal ischemia-reperfusion increases efflux for uric acid via paracellular route in the intestine, but decreases that via transcellular route mediated by BCRP., J Pharm Pharm Sci, 15(2) 295-304, 2012

    Ogura, Jiro Kuwayama, Kaori Takaya, Atsushi Terada, Yusuke Tsujimoto, Takashi Koizumi, Takahiro Maruyama, Hajime Fujikawa, Asuka Takahashi, Natsuko Kobayashi, Masaki Itagaki, Shirou Hirano, Takeshi Ya...

    Single Author

  • Intestinal Ischemia-Reperfusion Increases Efflux for Uric Acid Via Paracellular Route in the Intestine, but Decreases that Via Transcellular Route Mediated by BCRP, JOURNAL OF PHARMACY AND PHARMACEUTICAL SCIENCES, 15(2) 295-304, 2012

    Ogura, J; Kuwayama, K; Takaya, A; Terada, Y; Tsujimoto, T; Koizumi, T; Maruyama, H; Fujikawa, A; Takahashi, N; Kobayashi, M; Itagaki, S; Hirano, T; Yamaguchi, H; Iseki, K

    Single Author

  • The Decrease in Farnesoid X Receptor, Pregnane X Receptor and Constitutive Androstane Receptor in the Liver after Intestinal Ischemia-Reperfusion, JOURNAL OF PHARMACY AND PHARMACEUTICAL SCIENCES, 15(5) 616-631, 2012

    Ogura, J; Terada, Y; Tsujimoto, T; Koizumi, T; Kuwayama, K; Maruyama, H; Fujikawa, A; Takaya, A; Kobayashi, M; Itagaki, S; Takahashi, N; Hirano, T; Yamaguchi, H; Iseki, K

    Single Author

  • Quantification of intracellular and extracellular prostanoids stimulated by A23187 by liquid chromatography/electrospray ionization tandem mass spectrometry, JOURNAL OF CHROMATOGRAPHY B-ANALYTICAL TECHNOLOGIES IN THE BIOMEDICAL AND LIFE SCIENCES, 879(30) 3378-3385, 2011.11

    Furugen, A; Yamaguchi, H; Tanaka, N; Ito, H; Miyamori, K; Fujikawa, A; Takahashi, N; Ogura, J; Kobayashi, M; Yamada, T; Mano, N; Iseki, K

    Single Author

  • Effect of different surface treatments on the repair strength of a nanofilled resin-based composite, DENTAL MATERIALS JOURNAL, 30(4) 537-545, 2011.07

    Hamano, N; Chiang, YC; Nyamaa, I; Yamaguchi, H; Ino, S; Hickel, R; Kunzelmann, KH

    Single Author

  • An accurate quantitative LC/ESI-MS/MS method for sirolimus in human whole blood, JOURNAL OF CHROMATOGRAPHY B-ANALYTICAL TECHNOLOGIES IN THE BIOMEDICAL AND LIFE SCIENCES, 879(13-14) 987-992, 2011.04

    Mano, N; Sato, M; Nozawa, M; Matsumoto, Y; Mori, M; Yamaguchi, H; Goto, J; Shimada, M

    Single Author

  • Identification and elimination of ion suppression in the quantitative analysis of sirolimus in human blood by LC/ESI-MS/MS, JOURNAL OF CHROMATOGRAPHY B-ANALYTICAL TECHNOLOGIES IN THE BIOMEDICAL AND LIFE SCIENCES, 879(13-14) 968-974, 2011.04

    Mano, N; Nozawa, M; Sato, M; Mori, M; Yamaguchi, H; Kanda, K; Nogami, M; Goto, J; Shimada, M

    Single Author

  • Screening of Antibiotics That Interact with Organic Anion-Transporting Polypeptides 1B1 and 1B3 Using Fluorescent Probes, BIOLOGICAL & PHARMACEUTICAL BULLETIN, 34(3) 389-395, 2011.03

    Yamaguchi, H; Takeuchi, T; Okada, M; Kobayashi, M; Unno, M; Abe, T; Goto, J; Hishinuma, T; Shimada, M; Mano, N

    Single Author

  • FXR, PXR and CAR were Decreased in the Liver but not in the Jejunum after Intestinal Ischemia-reperfusion, DRUG METABOLISM REVIEWS, 42 277-278, 2010.08

    Jiro, O; Yusuke, T; Kobayashi, M; Itagaki, S; Yamaguchi, H; Iseki, K

    Single Author

  • Production of <SUP>18</SUP>O-Single Labeled Peptide Fragments during Trypsin Digestion of Proteins for Quantitative Proteomics Using nanoLC-ESI-MS/MS, JOURNAL OF PROTEOME RESEARCH, 9(7) 3741-3749, 2010.07

    Mori, M; Abe, K; Yamaguchi, H; Goto, J; Shimada, M; Mano, N

    Single Author

  • Transport of Estrone 3-sulfate Mediated by Organic Anion Transporter OATP4C1: Estrone 3-sulfate binds to the Different Recognition Site for Digoxin in OATP4C1, DRUG METABOLISM AND PHARMACOKINETICS, 25(3) 314-317, 2010

    Yamaguchi, H; Sugie, M; Okada, M; Mikkaichi, T; Toyohara, T; Abe, T; Goto, J; Hishinuma, T; Shimada, M; Mano, N

    Single Author

  • SLCO4C1 Transporter Eliminates Uremic Toxins and Attenuates Hypertension and Renal Inflammation, JOURNAL OF THE AMERICAN SOCIETY OF NEPHROLOGY, 20(12) 2546-2555, 2009.12

    Toyohara, T; Suzuki, T; Morimoto, R; Akiyama, Y; Souma, T; Shiwaku, HO; Takeuchi, Y; Mishima, E; Abe, M; Tanemoto, M; Masuda, S; Kawano, H; Maernura, K; Nakayama, M; Sato, H; Mikkaichi, T; Yamaguchi, ...

    Single Author

  • Analysis of Phosphorylated Peptides by Double Pseudoneutral Loss Extraction Coupled with Derivatization Using <i>N</i>-(4-Bromobenzoyl)aminoethanethiol, ANALYTICAL CHEMISTRY, 81(22) 9395-9401, 2009.11

    Mano, N; Aoki, S; Yamazaki, T; Nagaya, Y; Mori, M; Abe, K; Shimada, M; Yamaguchi, H; Goto, T; Goto, J

    Single Author

  • Introducing Hazard Prediction Training 'KYT' to Undergraduate Pharmacy Education on Patient Safety, YAKUGAKU ZASSHI-JOURNAL OF THE PHARMACEUTICAL SOCIETY OF JAPAN, 129(11) 1367-1373, 2009.11

    Murai, Y; Sato, M; Yamaguchi, H; Shimada, M; Mano, N; Goto, J; Hishinuma, T

    Single Author

  • Bonding strength of autopolymerizing resin to nylon denture base polymer, DENTAL MATERIALS JOURNAL, 28(4) 409-418, 2009.07

    Katsumata, Y; Hojo, S; Hamano, N; Watanabe, T; Yamaguchi, H; Okada, S; Teranaka, T; Ino, S

    Single Author

  • Contribution of the drug transporter ABCG2 (breast cancer resistance protein) to resistance against anticancer nucleosides, MOLECULAR CANCER THERAPEUTICS, 7(9) 3092-3102, 2008.09

    de Wolf, C; Jansen, R; Yamaguchi, H; de Haas, M; de Wetering, KV; Wijnholds, J; Beijnen, J; Borst, P

    Single Author

  • Simple quantification of lansoprazole and rabeprazole concentrations in human serum by liquid chromatography/tandem mass spectrometry, JOURNAL OF CHROMATOGRAPHY B-ANALYTICAL TECHNOLOGIES IN THE BIOMEDICAL AND LIFE SCIENCES, 870(1) 38-45, 2008.07

    Hishinuma, T; Suzuki, K; Yamaguchi, H; Yamagishi, H; Koike, T; Ohara, S; Shimosegawa, T; Mano, N; Goto, J

    Single Author

  • Rapid screening of antineoplastic candidates for the human organic anion transporter OATP1B3 substrates using fluorescent probes, CANCER LETTERS, 260(1-2) 163-169, 2008.02

    Yamaguchi, H; Kobayashi, M; Okada, M; Takeuchi, T; Unno, M; Abe, T; Goto, J; Hishinuma, T; Mano, N

    Single Author

  • Functional analysis of organic anion transporter, OATP4C1, expressed in kidney, YAKUGAKU ZASSHI-JOURNAL OF THE PHARMACEUTICAL SOCIETY OF JAPAN, 128 51-52, 2008

    Yamaguchi, H; Sugie, M; Okada, M; Abe, T; Goto, J; Hishinuma, T; Shimada, M; Mano, N

    Single Author

  • Simultaneous quantification of seven prostanoids using liquid chromatography/tandem mass spectrometry: The effects of arachidonic acid on prostanoid production in mouse bone marrow-derived mast cells, PROSTAGLANDINS LEUKOTRIENES AND ESSENTIAL FATTY ACIDS, 76(6) 321-329, 2007.06

    Hishinuma, T; Suzukia, K; Saitoa, M; Yamaguchi, H; Suzuki, N; Tomioka, Y; Kaneko, I; Ono, M; Goto, J

    Single Author

  • cGMP transport by vesicles from human and mouse erythrocytes, FEBS JOURNAL, 274(2) 439-450, 2007.01

    de Wolf, CJF; Yamaguchi, H; van der Heijden, I; Wielinga, PR; Hundscheid, SL; Ono, N; Scheffer, GL; de Haas, M; Schuetz, JD; Wijnholds, J; Borst, P

    Single Author

  • Study on the visualization of carrier-mediated transport, YAKUGAKU ZASSHI-JOURNAL OF THE PHARMACEUTICAL SOCIETY OF JAPAN, 127 181-182, 2007

    Okada, M; Yamaguchi, H; Kobayashi, M; Takeuchi, T; Tanemoto, M; Unno, M; Abe, T; Hishinuma, T; Goto, J; Mano, N

    Single Author

  • Transport of fluorescent chenodeoxycholic acid via the human organic anion transporters OATP1B1 and OATP1B3, JOURNAL OF LIPID RESEARCH, 47(6) 1196-1202, 2006.06

    Yamaguchi, H; Okada, M; Akitaya, S; Ohara, H; Mikkaichi, T; Ishikawa, H; Sato, M; Matsuura, M; Saga, T; Unno, M; Abe, T; Mano, N; Hishinuma, T; Goto, J

    Single Author

  • Utility of gallium-67 scintigraphy for evaluation of cardiac sarcoidosis with ventricular tachycardia, INTERNATIONAL JOURNAL OF CARDIOVASCULAR IMAGING, 22(3-4) 443-448, 2006.06

    Futamatsu, H; Suzuki, J; Adachi, S; Okada, H; Otomo, K; Ohara, T; Hashimoto, Y; Kakuta, T; Iesaka, Y; Yamaguchi, H; Sakurada, H; Sato, A; Obayashi, T; Niwa, A; Hirao, K; Isobe, M

    Single Author

  • Simultaneous determination of pancuronium, vecuronium and their related compounds using LC-ESI-MS., Leg Med (Tokyo), 8(3) 166-171, 2006.05

    Usui, Kiyotaka Hishinuma, Takanori Yamaguchi, Hiroaki Saga, Toshihide Wagatsuma, Toshihiro Hoshi, Kunihiko Tachiiri, Naoki Miura, Kuniaki Goto, Junichi

    Single Author

  • Genetic variation in <i>ABCB1</i> influences paclitaxel pharmacokinetics in Japanese patients with ovarian cancer, INTERNATIONAL JOURNAL OF GYNECOLOGICAL CANCER, 16(3) 979-985, 2006.05

    Yamaguchi, H; Hishinuma, T; Endo, N; Tsukamoto, H; Kishikawa, Y; Sato, M; Murai, Y; Hiratsuka, M; Ito, K; Okamura, C; Yaegashi, N; Suzuki, N; Tomioka, Y; Goto, J

    Single Author

  • Preparation of neocarzinostatin apoprotein mutants and the randomized library on the chromophore-binding cavity, BIOLOGICAL & PHARMACEUTICAL BULLETIN, 29(5) 1010-1014, 2006.05

    Tomioka, Y; Kisara, S; Yoshizawa, S; Ozawa, M; Suzuki, N; Yamaguchi, H; Hishinuma, T; Mizugaki, M; Goto, J

    Single Author

  • Determination of chlorhexidine (CHD) and nonylphenolethoxylates (NPEO<i>n</i>) using LC-ESI-MS method and application to hemolyzed blood, JOURNAL OF CHROMATOGRAPHY B-ANALYTICAL TECHNOLOGIES IN THE BIOMEDICAL AND LIFE SCIENCES, 831(1-2) 105-109, 2006.02

    Usui, K; Hishinuma, T; Yamaguchi, H; Tachiiri, N; Goto, J

    Single Author

  • Properties of asymmetric BPDA based phenylethynyl terminated thermosetting polyimide and its composite, JOURNAL OF PHOTOPOLYMER SCIENCE AND TECHNOLOGY, 19(2) 269-272, 2006

    Yamaguchi, H; Aoki, F

    Single Author

  • Effect of cisplatin-induced acute renal failure on bioavailability and intestinal secretion of quinolone antibacterial drugs in rats, PHARMACEUTICAL RESEARCH, 21(2) 330-338, 2004.02

    Yamaguchi, H; Yano, I; Saito, H; Inui, K

    Single Author

  • Pharmacokinetic role of P-glycoprotein in oral bioavailability and intestinal secretion of grepafloxacin in vivo, JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 300(3) 1063-1069, 2002.03

    Yamaguchi, H; Yano, I; Saito, H; Inui, KI

    Single Author

  • Transport characteristics of grepafloxacin and levofloxacin in the human intestinal cell line Caco-2, EUROPEAN JOURNAL OF PHARMACOLOGY, 431(3) 297-303, 2001.11

    Yamaguchi, H; Yano, I; Saito, H; Inui, KI

    Single Author

  • Secretory mechanisms of grepafloxacin and levofloxacin in the human intestinal cell line caco-2., J Pharmacol Exp Ther, 295(1) 360-366, 2000.10

    Yamaguchi, H Yano, I Hashimoto, Y Inui, K I

    Single Author

  • Secretory mechanisms of grepafloxacin and levofloxacin in the human intestinal cell line Caco-2, JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 295(1) 360-366, 2000.10

    Yamaguchi, H; Yano, I; Hashimoto, Y; Inui, KI

    Single Author

  • Microdetermination of the 6,15-diketo-13,14-dihydroprostaglandin F<sub>1α</sub> in human plasma using gas chromatography/selected ion monitoring with [<SUP>18</SUP>O]6,15-diketo-13,14-dihydro-prostaglandin F<sub>1α</sub> as an internal standard, PROSTAGLANDINS & OTHER LIPID MEDIATORS, 58(2-4) 187-193, 1999.10

    Mizugaki, M; Hishinuma, T; Yamaguchi, H; Kanno, K; Hirose, Y; Nakamura, H

    Single Author

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Review Papers

  • 薬学部病院実習における他職種業務見学プログラムの効果と課題, 医療薬学フォーラム講演要旨集, 31st , 2023

    小倉次郎, 志田敏宏, 畠山史朗, 山口浩明

  • プラチナ感受性再発卵巣がんに対するオラパリブのコンパニオン診断による薬剤経済評価, 日本癌治療学会学術集会抄録集, 57回 P157-6, 2019.10

    志田 敏宏, 佐藤 一真, 中村 達也, 山口 浩明, 荒川 一郎, 井上 忠夫

  • LC/ESI‐MS/MSを用いる胆汁酸メタボローム解析系の基礎的検討, (一社)日本臨床化学会, 臨床化学, 48(Suppl.1) 289, 2019.08

    庄子彩織, 前川正充, 山口浩明, 山口浩明, 眞野成康, 眞野成康

  • LC‐MS/MSを用いる脂質メディエーター網羅的解析の基礎的検討, (一社)日本臨床化学会, 臨床化学, 48(Suppl.1) 290, 2019.08

    横田真希, 前川正充, 福田隼, 眞野成康, 眞野成康, 山口浩明

  • LC/MS/MSによるニーマンピック病C型モデル細胞中ステロイドホルモン類の挙動解析, (一社)日本臨床化学会, 臨床化学, 48(Suppl.1) 289, 2019.08

    阿部愛, 前川正充, 小倉次郎, 山口浩明, 山口浩明, 眞野成康, 眞野成康

  • 血清リン脂質類のLC‐MS/MS分析に基づくニーマンピック病C型の迅速スクリーニング法の検討, (一社)日本臨床化学会, 臨床化学, 48(Suppl.1) 290, 2019.08

    岩堀杏南, 前川正充, 山口浩明, 眞野成康, 眞野成康

  • グローバルメタボロミクスによるニーマンピック病C型患者血液に特徴的なピーク探索, (一社)日本医用マススペクトル学会, JSBMS Letters, 44(Supplement) 79, 2019.08

    前川正充, 前川正充, 岩堀杏南, 金光祥臣, 三枝大輔, 三枝大輔, 山口浩明, 山口浩明, 山口浩明, 眞野成康, 眞野成康

  • 【がん治療と薬物相互作用 ピットフォールに陥らないための基礎と実践】抗がん薬の薬物動態学的 薬力学的相互作用 薬物動態学的機序による抗がん薬の薬物相互作用, (株)南山堂, 薬局, 70(7) 1425-1431, 2019.06

    山口 浩明, 菊地 正史

  • 第2回病院薬剤師が実践するリバーストランスレーショナルリサーチの最前線〜分子標的探索と個別化医療への挑戦〜 経口分子標的薬の個別化投与設計に向けて, (公社)日本薬学会, 薬学雑誌, 139(6) 911-915, 2019.06

    山口 浩明, 高崎 新也, 菊地 正史, 川崎 芳英, 荒井 陽一, 眞野 成康

  • 血中エベロリムス濃度と臨床効果の関連性~腎癌治療における長期追跡調査~, TDM研究, 36(2) 138, 2019.05

    高崎新也, 川崎芳英, 菊地正史, 田中雅樹, 山口浩明, 伊藤明宏, 眞野成康

  • 経口がん分子標的薬の個別投与設計に向けた取り組み, 日本薬剤学会年会講演要旨集(Web), 34年会 34, 2019.05

    山口浩明, 高崎新也, 菊地正史, 川崎芳英, 伊藤明宏, 眞野成康

  • 日本人肺移植患者におけるミコフェノール酸およびミコフェノール酸アシルグルクロン酸抱合体のAUC0-12の推定式, (一社)日本TDM学会, TDM研究, 36(2) 135, 2019.05

    田中 雅樹, 菊地 正史, 高崎 新也, 野田 あおい, 秋場 美紀, 松田 安史, 大石 久, 野田 雅史, 岡田 克典, 眞野 成康, 山口 浩明

  • インソースCIDを利用したLC/ESI-MS/MSによる多種薬物の同時測定法の構築に向けた基礎検討, (公社)日本薬学会, 日本薬学会年会要旨集, 139年会(4) 114, 2019.03

    佐藤 裕, 前川 正充, 塚本 多矩, 高崎 新也, 菊地 正史, 早川 禎宏, 山口 浩明, 眞野 成康

  • Toward Personalized Cancer Therapy with Oral Molecular-targeted Agents, 薬学雑誌(Web), 139(6) 911‐915(J‐STAGE), 2019

    山口浩明, 高崎新也, 菊地正史, 川崎芳英, 荒井陽一, 眞野成康

  • LC/ESI‐MS/MSを用いるニーマンピック病C型モデル細胞のステロイドホルモン代謝解析, 日本薬学会年会要旨集(CD-ROM), 139th(2) ROMBUNNO.23PO‐am151-274, 2019

    阿部愛, 前川正充, 小倉次郎, 須賀隆浩, 檜垣克己, 山口浩明, 山口浩明, 山口浩明, 眞野成康, 眞野成康, 眞野成康

  • スニチニブのTDM普及に向けて, 日本臨床腫瘍薬学会学術大会講演要旨集, 2019 138, 2019

    山口浩明, 高崎新也, 菊地正史, 川崎芳英, 荒井陽一, 眞野成康

  • 腎癌治療における日本人のスニチニブ血中濃度と有害事象の関連性評価, 日本臨床腫瘍薬学会学術大会講演要旨集, 2019 151, 2019

    高崎新也, 川崎芳英, 菊地正史, 田中雅樹, 細野寛貴, 伊藤明宏, 山口浩明, 眞野成康

  • 中毒起因物質の実用的分析法 カルシウム拮抗剤の分析, (株)へるす出版, 中毒研究, 31(3) 302-307, 2018.09

    安藤 基純, 有吉 孝一, 臼井 聖尊, 斉藤 剛, 藤田 友嗣, 堀 寧, 三瀬 雅史, 山口 浩明, 芳澤 朋大, 日本中毒学会分析委員会

  • 治療効果の最大化を目指した経口抗がん薬の治療薬物モニタリング, JSBMS Letters, 43(Supplement) 49, 2018.08

    高崎新也, 川崎芳英, 菊地正史, 田中雅樹, 山口浩明, 眞野成康

  • 臨床化学研究における質量分析の貢献 治療効果の最大化を目指した経口抗がん薬の治療薬物モニタリング, (一社)日本医用マススペクトル学会, JSBMS Letters, 43(Suppl.) 49, 2018.08

    高崎 新也, 川崎 芳英, 菊地 正史, 田中 雅樹, 山口 浩明, 眞野 成康

  • LC/ESI-MS/MSを用いるコレステロール代謝物網羅的解析法の基礎的検討, (一社)日本臨床化学会, 臨床化学, 47(Suppl.1) 320, 2018.07

    前川 正充, 河俣 圭太, 阿部 愛, 三枝 大輔, 山口 浩明, 眞野 成康

  • 薬学研究が支える臨床化学 臨床化学を基盤とした肺移植患者の個別化薬物療法構築への取り組み, (一社)日本臨床化学会, 臨床化学, 47(Suppl.1) 204, 2018.07

    菊地 正史, 山口 浩明, 眞野 成康

  • 質量分析の活用事例とピットフォール 個別化医療における血中薬物濃度の精密測定, (一社)日本臨床化学会, 臨床化学, 47(Suppl.1) 179, 2018.07

    眞野 成康, 前川 正充, 菊地 正史, 山口 浩明

  • 肺移植患者における個別化薬物療法, (公財)臨床薬理研究振興財団, 臨床薬理の進歩, (39) 104-116, 2018.06

    山口 浩明, 菊地 正史, 田中 雅樹, 高崎 新也, 野田 あおい, 重田 健介, 白木 美香, 高木 秀侑, 松田 安史, 野田 雅史, 岡田 克典, 眞野 成康

  • インソースCIDを利用したLC/ESI-MS/MSによるチロシンキナーゼ阻害薬一斉測定法の構築, (公社)日本薬学会, 日本薬学会年会要旨集, 138年会(4) 175, 2018.03

    佐藤 裕, 高崎 新也, 田中 雅樹, 前川 正充, 菊地 正史, 川崎 芳英, 荒井 陽一, 山口 浩明, 眞野 成康

  • レセプトデータを利用した小児ADHD患者における処方実態の把握, (公社)日本薬学会, 日本薬学会年会要旨集, 138年会(4) 185, 2018.03

    吉田 真貴子, 小原 拓, 菊地 紗耶, 菊地 正史, 山口 浩明, 眞野 成康

  • 第2回臨床化学の進歩が変える薬物治療〜臨床病態解析からのアプローチ〜 オミクス解析を基盤とした臨床化学分析, (公社)日本薬学会, 日本薬学会年会要旨集, 138年会(1) 174, 2018.03

    眞野 成康, 前川 正充, 山口 浩明

  • 第2回病院薬剤師が実践するリバーストランスレーショナルリサーチの最前線〜分子標的探索と個別化医療への挑戦〜 経口分子標的薬の個別化投与設計に向けて, (公社)日本薬学会, 日本薬学会年会要旨集, 138年会(1) 134, 2018.03

    山口 浩明, 高崎 新也, 菊地 正史, 川崎 芳英, 荒井 陽一, 眞野 成康

  • アキシチニブにより薬剤性破壊性甲状腺炎を呈した腎癌患者の一例, 日本臨床腫瘍薬学会学術大会講演要旨集, 2018 183, 2018

    鈴鹿雅人, 高崎新也, 川崎芳英, 坪井真友子, 佐藤祐司, 山口浩明, 荒井陽一, 眞野成康

  • 臨床化学を基盤としたニーマンピック病C型の診断・治療への挑戦, 日本医療薬学会年会講演要旨集(Web), 28 , 2018

    前川正充, 成田綾, 崎山快夫, 山口浩明, 眞野成康

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Grant-in-Aid for Scientific Research

  • Grant-in-Aid for Scientific Research(C),2023.04 - 2026.03

  • Grant-in-Aid for Scientific Research(C),2022.04 - 2026.03

Other external funds procured

  • Participation of OATP4C1 in the pharmacokinetics of drugs,2018.04 - 2021.03,Participation of OATP4C1 in the pharmacokinetics of drugs

    Japan Society for the Promotion of Science

  • Medicinal chemistry studies based on the three-dimensional structural diversity-oriented molecular design of pharmacologically active compounds,2015.04 - 2020.03,Medicinal chemistry studies based on the three-dimensional structural diversity-oriented molecular design of pharmacologically active compounds

    Based on the three-dimensional structural diversity-oriented strategy using characteristic structural features of cyclopropane, medicinal chemistry studies have been carried out. As the result of these studies, various pharmacologically active compounds, such as, highly active congeners of pro-resolving lipid mediator RvE2, peptidomimetics including prorenin inhibitors and melanocortin receptor-4 selective ligands, membrane-permeable cyclic peptides, or the first GABA transporter GAT1-selective inhibitor, were identified. Thus, it was demonstrated that the three-dimensional structural diversity-oriented strategy effectively works for the theoretical development of desired pharmacologically active compounds. In addition, various synthetic procedures for the substituted chiral cyclopropanes, which can be effectively used in cyclopropane medicinal chemistry studies, have been developed.

    Japan Society for the Promotion of Science

Presentations

  • 臨床化学, Domestic presentation, 2019.08, 血清リン脂質類のLC‐MS/MS分析に基づくニーマンピック病C型の迅速スクリーニング法の検討, Oral presentation (general)

  • 臨床化学, Domestic presentation, 2019.08, LC/ESI‐MS/MSを用いる胆汁酸メタボローム解析系の基礎的検討, Oral presentation (general)

  • 臨床化学, Domestic presentation, 2019.08, LC‐MS/MSを用いる脂質メディエーター網羅的解析の基礎的検討, Oral presentation (general)

  • TDM研究, Domestic presentation, 2019.05, 血中エベロリムス濃度と臨床効果の関連性~腎癌治療における長期追跡調査~, Oral presentation (general)

  • 日本薬学会年会要旨集(CD-ROM), Domestic presentation, 2019, LC/ESI‐MS/MSを用いるニーマンピック病C型モデル細胞のステロイドホルモン代謝解析, Oral presentation (general)

  • 日本臨床腫瘍薬学会学術大会講演要旨集, Domestic presentation, 2019, 腎癌治療における日本人のスニチニブ血中濃度と有害事象の関連性評価, Oral presentation (general)

  • 日本薬剤学会年会講演要旨集(Web), Domestic presentation, 2019, 経口がん分子標的薬の個別投与設計に向けた取り組み, Symposium, workshop panel (public)

  • 日本臨床腫瘍薬学会学術大会講演要旨集, Domestic presentation, 2019, スニチニブのTDM普及に向けて, Symposium, workshop panel (public)

  • 日本臨床腫瘍薬学会学術大会講演要旨集, Domestic presentation, 2018, アキシチニブにより薬剤性破壊性甲状腺炎を呈した腎癌患者の一例, Oral presentation (general)

  • 日本先天代謝異常学会雑誌, Domestic presentation, 2017.09, 5種の尿中抱合型代謝物をマルチバイオマーカーとして用いるニーマンピック型C型の化学診断法の開発, Oral presentation (general)

  • 臨床化学, Domestic presentation, 2017.09, 尿中アシルカルニチンの一斉定量法の構築, Oral presentation (general)

  • 臨床化学, Domestic presentation, 2017.09, UHPLC-UVによるエルロチニブ及び代謝物の同時測定法と非小細胞肺がん患者血中濃度測定への応用, Oral presentation (general)

  • 臨床化学, Domestic presentation, 2017.09, PETINIAとLC-MS/MSで得られた肺移植患者のミコフェノール酸血中濃度の比較, Oral presentation (general)

  • 臨床化学, Domestic presentation, 2017.09, LC/ESI-MS/MSを用いたシロリムスの全血中濃度測定法の構築, Oral presentation (general)

  • 日本泌尿器科学会総会, Domestic presentation, 2017.04, スニチニブ投与により4年間完全奏功が維持できた腎細胞癌患者1症例のスニチニブ血中濃度推移, Oral presentation (general)

  • 日本薬学会年会要旨集, Domestic presentation, 2017.03, LC/ESI-MS/MSを用いた薬毒物中毒原因物質迅速スクリーニングの有用性, Oral presentation (general)

  • 日本臨床腫瘍薬学会学術大会講演要旨集, Domestic presentation, 2017, 外来治療中に経口抗がん薬の血中濃度測定により服薬アドヒアランスが向上した2例, Oral presentation (general)

  • 日本癌治療学会学術集会抄録集, Domestic presentation, 2016.10, 腎 腎がん分子標的治療の現況 切除不能腎癌治療におけるSunitinibの至適血中濃度の検討, Oral presentation (general)

  • 日本泌尿器科学会総会, Domestic presentation, 2016.04, 日本人の腎細胞癌患者におけるスニチニブの有効血中濃度域の検討, Oral presentation (general)

  • 日本生化学会大会・日本分子生物学会年会合同大会講演要旨集, Domestic presentation, 2015.12, 肝臓におけるhypoxia-inducible factor 1αの活性化はコレステロール胆石形成を促進する, Oral presentation (general)

  • 日本医療薬学会年会講演要旨集, Domestic presentation, 2015.10, アキシチニブの血中濃度が上昇しなかった腎細胞癌患者の一例, Oral presentation (general)

  • 日本医薬品情報学会総会・学術大会講演要旨集, Domestic presentation, 2014.07, 医薬品リスク管理計画に関する薬剤師の認識, Oral presentation (general)

  • 日本薬学会年会要旨集(CD-ROM), Domestic presentation, 2014, ダプトマイシンは骨格筋細胞におけるモノカルボン酸輸送担体の発現を低下させる, Oral presentation (general)

  • 日本医薬品情報学会総会・学術大会講演要旨集, Domestic presentation, 2013.08, 薬剤師における医薬品安全性評価に関する認識および実践に関する調査, Oral presentation (general)

  • 日本薬学会年会要旨集(CD-ROM), Domestic presentation, 2013, 抗MRSA薬ダプトマイシンの骨格筋細胞毒性に関する基礎的検討, Oral presentation (general)

  • Chromatography, Domestic presentation, 2011.10, Quantitation of antineoplastic drug oxaliplatin from human plasma using HILIC/MS/MS, Oral presentation (general)

  • 日本医療薬学会年会講演要旨集, Domestic presentation, 2011.09, PKCを介した糖代謝制御およびMCT4発現変動への関連性, Oral presentation (general)

  • 日本薬学会年会要旨集, Domestic presentation, 2011.03, ABCトランスポーター発現変動と酸化障害の重度との関連, Oral presentation (general)

  • 日本薬学会年会要旨集, Domestic presentation, 2011.03, 抗菌薬アミカシンの用法用量別にみた治療効果の比較, Oral presentation (general)

  • 日本薬学会年会要旨集, Domestic presentation, 2011.03, カラムスイッチング‐LC/MS/MSによるパクリタキセル血中濃度測定法の確立, Oral presentation (general)

  • 移植, Domestic presentation, 2007.06, 当院における膵島移植後の免疫抑制剤シロリムス血中濃度測定(LC/ESI‐MS/MSとMEIAの有用性について), Oral presentation (general)

  • 日本薬学会年会要旨集, Domestic presentation, 2007.03, LC/ESI‐MS/MS法およびIMx法による免疫抑制剤シロリムスの血中濃度測定, Oral presentation (general)

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